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Approval Year

Substance Class Protein
Created
by admin
on Mon Oct 21 20:41:07 UTC 2019
Edited
by admin
on Mon Oct 21 20:41:07 UTC 2019
Protein Sub Type
Sequence Type COMPLETE
Record UNII
6NP3XSMIP3
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MULTIDRUG AND TOXIN EXTRUSION PROTEIN 1
Common Name English
MATE1
Common Name English
FLJ10847
Common Name English
SOLUTE CARRIER FAMILY 47 MEMBER 1
Common Name English
SLC47A1
Common Name English
MGC64822
Common Name English
MATE-1
Common Name English
Classification Tree Code System Code
UCSF-FDA TRANSPORTAL SLC47A1
Created by admin on Mon Oct 21 20:41:07 UTC 2019 , Edited by admin on Mon Oct 21 20:41:07 UTC 2019
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Rifamycin is an inhibitor of renal transporters organic anion transporter (OAT) 3, multidrug and toxin extrusion (MATE) 1, and MATE2-K transporters in vitro, however, based on systemic concentrations of rifamycin observed after administration of the recommended dose, clinically relevant inhibition of these transporters in vivo is unlikely.
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INHIBITOR -> METABOLIC ENZYME
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INHIBITOR -> TRANSPORTER
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WEAK
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SUBSTRATE -> TRANSPORTER
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Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL