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Development Status
Investigational
148
US Approved Rx
32
Possibly Marketed Outside US
2
US Previously Marketed
1
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Primary Target
Receptor tyrosine-protein kinase erbB-2
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Approved
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Approval Year
Unknown
149
2015
5
2014
4
2004
3
2019
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Condition
Breast cancer
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Treatment Modality
Primary
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Originator
Genentech
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Substance Class
Protein
147
Concept
27
Structurally Diverse
5
Nucleic Acid
4
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Code System
FDA UNII
183
NCI_THESAURUS
183
CAS
159
INN
152
USAN
117
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Protein Type
MONOCLONAL ANTIBODY
125
MONOCLONAL ANTIBODY CONJUGATE
12
BISPECIFIC ANTIBODY
7
BISPECIFIC MONOCLONAL FRAGMENTS
1
MONOCLONAL ANTIBODY FUSION PROTEIN
1
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ATC Level 1
ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS
25
MUSCULO-SKELETAL SYSTEM
1
NERVOUS SYSTEM
1
VARIOUS
1
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ATC Level 2
ANTINEOPLASTIC AGENTS
22
IMMUNOSUPPRESSANTS
4
DRUGS FOR TREATMENT OF BONE DISEASES
1
OTHER NERVOUS SYSTEM DRUGS
1
THERAPEUTIC RADIOPHARMACEUTICALS
1
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ATC Level 3
OTHER ANTINEOPLASTIC AGENTS
22
IMMUNOSUPPRESSANTS
4
DRUGS AFFECTING BONE STRUCTURE AND MINERALIZATION
1
OTHER NERVOUS SYSTEM DRUGS
1
OTHER THERAPEUTIC RADIOPHARMACEUTICALS
1
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ATC Level 4
Monoclonal antibodies
21
Interleukin inhibitors
2
Selective immunosuppressants
2
Iodine (<sup>131</sup>I) compounds
1
Other antineoplastic agents
1
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Substance Form
Principal Form
182
Salts, Hydrates, Esters, etc.
1
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Search results for
"Pharmacologic Substance[C1909]|Biological Agent[C307]|Antineoplastic Biological Agent"
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TISOTUMAB VEDOTIN
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T41737F88A
Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
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Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Status:
US Approved Rx (2021)
First approved in 2021
Class:
PROTEIN
SACITUZUMAB GOVITECAN
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M9BYU8XDQ6
Subunit
1
(451) Similarity Search
Subunit
2
(451) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Export Data
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Subunit
1
(451) Similarity Search
Subunit
2
(451) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Status:
US Approved Rx (2020)
First approved in 2020
Class:
PROTEIN
TEPROTUMUMAB
MORE DETAILS
Y64GQ0KC0A
Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(215) Similarity Search
Subunit
4
(215) Similarity Search
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Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(215) Similarity Search
Subunit
4
(215) Similarity Search
Status:
US Approved Rx (2020)
First approved in 2020
Class:
PROTEIN
TRASTUZUMAB DERUXTECAN
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5384HK7574
Subunit
1
(450) Similarity Search
Subunit
2
(450) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Export Data
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Subunit
1
(450) Similarity Search
Subunit
2
(450) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Status:
US Approved Rx (2019)
First approved in 2019
Class:
PROTEIN
ENFORTUMAB VEDOTIN
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DLE8519RWM
Subunit
1
(447) Similarity Search
Subunit
2
(447) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
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Subunit
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(447) Similarity Search
Subunit
2
(447) Similarity Search
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3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Status:
US Approved Rx (2019)
First approved in 2019
Class:
PROTEIN
POLATUZUMAB VEDOTIN
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KG6VO684Z6
Subunit
1
(447) Similarity Search
Subunit
2
(447) Similarity Search
Subunit
3
(218) Similarity Search
Subunit
4
(218) Similarity Search
Export Data
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Subunit
1
(447) Similarity Search
Subunit
2
(447) Similarity Search
Subunit
3
(218) Similarity Search
Subunit
4
(218) Similarity Search
Status:
US Approved Rx (2019)
First approved in 2019
Class:
PROTEIN
CEMIPLIMAB
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6QVL057INT
Subunit
1
(444) Similarity Search
Subunit
2
(444) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
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(444) Similarity Search
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2
(444) Similarity Search
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(214) Similarity Search
Subunit
4
(214) Similarity Search
Status:
US Approved Rx (2018)
First approved in 2018
Class:
PROTEIN
GUSELKUMAB
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089658A12D
Subunit
1
(446) Similarity Search
Subunit
2
(446) Similarity Search
Subunit
3
(217) Similarity Search
Subunit
4
(217) Similarity Search
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(446) Similarity Search
Subunit
2
(446) Similarity Search
Subunit
3
(217) Similarity Search
Subunit
4
(217) Similarity Search
Status:
US Approved Rx (2017)
First approved in 2017
Class:
PROTEIN
INOTUZUMAB OZOGAMICIN
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P93RUU11P7
Subunit
1
(446) Similarity Search
Subunit
2
(446) Similarity Search
Subunit
3
(219) Similarity Search
Subunit
4
(219) Similarity Search
Export Data
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Subunit
1
(446) Similarity Search
Subunit
2
(446) Similarity Search
Subunit
3
(219) Similarity Search
Subunit
4
(219) Similarity Search
Status:
US Approved Rx (2017)
First approved in 2017
Class:
PROTEIN
OLARATUMAB
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TT6HN20MVF
Subunit
1
(457) Similarity Search
Subunit
2
(457) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
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Subunit
1
(457) Similarity Search
Subunit
2
(457) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Status:
US Approved Rx (2016)
First approved in 2016
Class:
PROTEIN
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