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NCATS
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Development Status
Investigational
144
US Approved Rx
37
Possibly Marketed Outside US
1
US Previously Marketed
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Primary Target
Receptor tyrosine-protein kinase erbB-2
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Approval Year
Unknown
145
2015
5
2014
4
2024
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2004
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Condition
Breast cancer
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Primary
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Originator
Genentech
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Substance Class
Protein
148
Concept
26
Structurally Diverse
5
Nucleic Acid
4
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Code System
FDA UNII
183
NCI_THESAURUS
183
SMS_ID
169
CAS
159
INN
152
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Protein Type
MONOCLONAL ANTIBODY
126
MONOCLONAL ANTIBODY CONJUGATE
12
BISPECIFIC ANTIBODY
7
BISPECIFIC MONOCLONAL FRAGMENTS
1
MONOCLONAL ANTIBODY FUSION PROTEIN
1
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ATC Level 1
ANTINEOPLASTIC AND IMMUNOMODULATING AGENTS
25
MUSCULO-SKELETAL SYSTEM
1
NERVOUS SYSTEM
1
VARIOUS
1
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ATC Level 2
ANTINEOPLASTIC AGENTS
22
IMMUNOSUPPRESSANTS
4
DRUGS FOR TREATMENT OF BONE DISEASES
1
OTHER NERVOUS SYSTEM DRUGS
1
THERAPEUTIC RADIOPHARMACEUTICALS
1
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ATC Level 3
OTHER ANTINEOPLASTIC AGENTS
22
IMMUNOSUPPRESSANTS
4
DRUGS AFFECTING BONE STRUCTURE AND MINERALIZATION
1
OTHER NERVOUS SYSTEM DRUGS
1
OTHER THERAPEUTIC RADIOPHARMACEUTICALS
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ATC Level 4
Monoclonal antibodies
21
Interleukin inhibitors
2
Selective immunosuppressants
2
Iodine (<sup>131</sup>I) compounds
1
Other antineoplastic agents
1
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Substance Form
Principal Form
182
Salts, Hydrates, Esters, etc.
1
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Search results for
"Pharmacologic Substance[C1909]|Biological Agent[C307]|Antineoplastic Biological Agent"
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Zolbetuximab
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TF5MPQ8WGY
Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(220) Similarity Search
Subunit
4
(220) Similarity Search
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Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(220) Similarity Search
Subunit
4
(220) Similarity Search
Status:
US Approved Rx (2024)
First approved in 2024
Class:
PROTEIN
Cosibelimab
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PNW7GBB44P
Subunit
1
(450) Similarity Search
Subunit
2
(450) Similarity Search
Subunit
3
(218) Similarity Search
Subunit
4
(218) Similarity Search
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Subunit
1
(450) Similarity Search
Subunit
2
(450) Similarity Search
Subunit
3
(218) Similarity Search
Subunit
4
(218) Similarity Search
Status:
US Approved Rx (2024)
First approved in 2024
Class:
PROTEIN
TISLELIZUMAB
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0KVO411B3N
Subunit
1
(445) Similarity Search
Subunit
2
(445) Similarity Search
Subunit
3
(214) Similarity Search
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(445) Similarity Search
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(445) Similarity Search
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(214) Similarity Search
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4
(214) Similarity Search
Status:
US Approved Rx (2024)
First approved in 2024
Class:
PROTEIN
Zenocutuzumab
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AE72RB1W1X
Subunit
1
(453) Similarity Search
Subunit
2
(450) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
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(453) Similarity Search
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(450) Similarity Search
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(214) Similarity Search
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(214) Similarity Search
Status:
US Approved Rx (2024)
First approved in 2024
Class:
PROTEIN
TISOTUMAB VEDOTIN
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T41737F88A
Subunit
1
(448) Similarity Search
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(214) Similarity Search
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(448) Similarity Search
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4
(214) Similarity Search
Status:
US Approved Rx (2021)
First approved in 2021
Class:
PROTEIN
SACITUZUMAB GOVITECAN
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M9BYU8XDQ6
Subunit
1
(451) Similarity Search
Subunit
2
(451) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
Export Data
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Subunit
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(451) Similarity Search
Subunit
2
(451) Similarity Search
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3
(214) Similarity Search
Subunit
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(214) Similarity Search
Status:
US Approved Rx (2020)
First approved in 2020
Class:
PROTEIN
TEPROTUMUMAB
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Y64GQ0KC0A
Subunit
1
(448) Similarity Search
Subunit
2
(448) Similarity Search
Subunit
3
(215) Similarity Search
Subunit
4
(215) Similarity Search
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(448) Similarity Search
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(215) Similarity Search
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(215) Similarity Search
Status:
US Approved Rx (2020)
First approved in 2020
Class:
PROTEIN
TRASTUZUMAB DERUXTECAN
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5384HK7574
Subunit
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Subunit
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(214) Similarity Search
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(214) Similarity Search
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(450) Similarity Search
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(214) Similarity Search
Status:
US Approved Rx (2019)
First approved in 2019
Class:
PROTEIN
ENFORTUMAB VEDOTIN
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DLE8519RWM
Subunit
1
(447) Similarity Search
Subunit
2
(447) Similarity Search
Subunit
3
(214) Similarity Search
Subunit
4
(214) Similarity Search
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(447) Similarity Search
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(447) Similarity Search
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(214) Similarity Search
Status:
US Approved Rx (2019)
First approved in 2019
Class:
PROTEIN
POLATUZUMAB VEDOTIN
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KG6VO684Z6
Subunit
1
(447) Similarity Search
Subunit
2
(447) Similarity Search
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3
(218) Similarity Search
Subunit
4
(218) Similarity Search
Export Data
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Subunit
1
(447) Similarity Search
Subunit
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(447) Similarity Search
Subunit
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(218) Similarity Search
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(218) Similarity Search
Status:
US Approved Rx (2019)
First approved in 2019
Class:
PROTEIN
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