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Approval Year

Unknown
127998
Substance Class Protein
Created
by admin
on Sun Dec 18 08:25:56 UTC 2022
Edited
by admin
on Sun Dec 18 08:25:56 UTC 2022
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
V23K99CV7G
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MUSCARINIC ACETYLCHOLINE RECEPTOR M1
Common Name English
CHRM1
Common Name English
Code System Code Type Description
PHAROS
P11229
Created by admin on Sun Dec 18 08:25:59 UTC 2022 , Edited by admin on Sun Dec 18 08:25:59 UTC 2022
PRIMARY
FDA UNII
V23K99CV7G
Created by admin on Sun Dec 18 08:25:59 UTC 2022 , Edited by admin on Sun Dec 18 08:25:59 UTC 2022
PRIMARY
UNIPROT
P11229
Created by admin on Sun Dec 18 08:25:59 UTC 2022 , Edited by admin on Sun Dec 18 08:25:59 UTC 2022
PRIMARY
From To
1_98 1_178
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_2
N 1_12
Related Record Type Details
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Structure of CYCLOPENTOLATE
INHIBITOR -> TARGET
Structure of SUCCINYLCHOLINE
AGONIST -> TARGET
Structure of TRIHEXYPHENIDYL
INHIBITOR -> TARGET
Structure of AZD-6088
PARTIAL AGONIST->TARGET
Structure of Aroxybutynin
INHIBITOR -> TARGET
Structure of NERATINIB
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Radioligand binding assay
BINDING
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Structure of ACLIDINIUM
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Structure of THRX-195518
INHIBITOR -> TARGET
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BINDING
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Structure of SOLIFENACIN
INHIBITOR -> TARGET
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Structure of TAK-071
POSITIVE ALLOSTERIC MODULATOR->TARGET
Structure of Pilocarpine
AGONIST -> TARGET
Structure of PALIPERIDONE
NON-INHIBITOR->OFF TARGET
NON-INHIBITOR
Ki
Structure of REVEFENACIN
INHIBITOR -> TARGET
BINDING
Kd
Structure of CARBACHOL
AGONIST -> TARGET
Structure of Oxybutynin
INHIBITOR -> TARGET
Structure of NERATINIB
INHIBITOR->OFF-TARGET
DOXEPIN
INHIBITOR -> TARGET
Structure of RISPERIDONE
NON-INHIBITOR->OFF TARGET
Ki
Structure of NORQUETIAPINE
INHIBITOR -> TARGET
Ki
Structure of ALVAMELINE
AGONIST -> TARGET
Structure of REVOSIMELINE
AGONIST -> TARGET
Structure of BLARCAMESINE
MODULATOR->TARGET
Structure of ATROPINE
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
NIH
NCATS
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