U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 03:49:08 GMT 2025
Edited
by admin
on Wed Apr 02 03:49:08 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
VZX139UJO5
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ADRB2
Preferred Name English
BETA-2 ADRENERGIC RECEPTOR
Common Name English
?2 adrenergic receptor
Common Name English
Beta-2 adrenoceptor
Common Name English
beta2
Common Name English
B2AR
Common Name English
BETA-2 ADRENORECEPTOR
Common Name English
ADRB2R
Common Name English
Code System Code Type Description
FDA UNII
VZX139UJO5
Created by admin on Wed Apr 02 03:49:08 GMT 2025 , Edited by admin on Wed Apr 02 03:49:08 GMT 2025
PRIMARY
UNIPROT
P07550
Created by admin on Wed Apr 02 03:49:08 GMT 2025 , Edited by admin on Wed Apr 02 03:49:08 GMT 2025
PRIMARY
From To
1_106 1_191
1_184 1_190
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_6
N 1_15
Related Record Type Details
AGONIST -> TARGET
EC50
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
RADIOLIGAND->TARGET
Used for cardiac PET adrenoreceptor imaging studies
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
RADIOLIGAND->TARGET
Used for cardiac PET adrenoreceptor imaging studies
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
In spontaneous tone isolated trachea
EC50
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
INHIBITOR -> TARGET
AGONIST -> TARGET
SHORT-ACTING
INHIBITOR -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
RADIOLIGAND->TARGET
Chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable levels.
Kd
RADIOLIGAND->TARGET
BINDING
Kd
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
INHIBITOR -> TARGET
Chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable levels.
Kd
AGONIST -> TARGET
SHORT-ACTING
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
Ki
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
NON-SELECTIVE
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
BINDING
Kd
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
SHORT-ACTING
AGONIST -> TARGET
SHORT-ACTING
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
non-selective beta blocker
ANTAGONIST->TARGET
Levobunolol (LB) is the levo-rotatory isomer of bunolol, a potent, nonselective antagonist of beta-adrenergic receptors.
AGONIST -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL