Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Sat Jun 26 16:51:35 UTC 2021
by
admin
on
Sat Jun 26 16:51:35 UTC 2021
|
Protein Type | RECEPTOR |
Protein Sub Type | REUPTAKE RECEPTOR |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
CJZ26L1EGI
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
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CJZ26L1EGI
Created by
admin on Sat Jun 26 16:51:39 UTC 2021 , Edited by admin on Sat Jun 26 16:51:39 UTC 2021
|
PRIMARY |
From | To |
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1_200 | 1_209 |
Glycosylation Type | HUMAN |
Glycosylation Link Type | Site |
---|---|
N | 1_208 |
N | 1_217 |
Related Record | Type | Details | ||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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LIGAND->TRANSPORTER | |||
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INHIBITOR -> TARGET |
IN-VITRO
IC50
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ANTAGONIST->TARGET |
Ki
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
(+)-Tramadol inhibits serotonin reuptake
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SUBSTRATE -> TRANSPORTER |
STIMULATES SEROTONIN RELEASE.
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SUBSTRATE -> TRANSPORTER |
Our data show that drugs known or suspected to increase the risk of PPH (eg, aminorex, fenfluramine, and chlorphentermine) are 5-HT transporter substrates, whereas drugs that have not been shown to increase the risk of PPH are less potent in this regard.
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TARGET |
Kd
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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LIGAND->BINDER | |||
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INHIBITOR -> TARGET | |||
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TARGET->RADIOLIGAND | |||
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INHIBITOR -> TRANSPORTER |
IN-VITRO
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RADIOLIGAND->TARGET |
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
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Molecular Formula | CHEMICAL |
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MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
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