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Showing 1 - 10 of 36 results

Status:
US Approved Rx (2006)
First approved in 2000

Class (Stereo):
CHEMICAL (ACHIRAL)



Meloxicam (brand name Mobic) is an nonsteroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Mobic is indicated for the relief of the signs and symptoms of osteoarthritis and rheumatoid arthritis, and has been available i...
Status:
US Approved Rx (2024)
First approved in 1988

Class (Stereo):
CHEMICAL (RACEMIC)



Nicardipine is a potent calcium channel blockader with marked vasodilator action used to treat high blood pressure and angina. By deforming the channel, inhibiting ion-control gating mechanisms, and/or interfering with the release of calcium from the...
Status:
US Approved Rx (2017)
First approved in 1982

Class (Stereo):
CHEMICAL (ACHIRAL)



Piroxicam is in a class of drugs called nonsteroidal anti-inflammatory drugs (NSAIDs). It was originally brought to market by Pfizer under the tradename Feldene in 1980, became generic in 1992, and is marketed worldwide under many brandnames. Piroxic...
Status:
US Approved Rx (1991)
First approved in 1978

Class (Stereo):
CHEMICAL (RACEMIC)



Sulindac is a nonsteroidal anti-inflammatory agent (NSAIA) of the arylalkanoic acid class that is marketed in the U.S. by Merck as Clinoril. Like other NSAIAs, it may be used in the treatment of acute or chronic inflammatory conditions. Sulindac is a...
Status:
US Approved Rx (1985)
First marketed in 1921

Class (Stereo):
CHEMICAL (ACHIRAL)



Pentaerythritol tetranitrate is an organic nitrate that has been used for the treatment of angina pectoris. Upon administration, the drug undergoes exstensive metabolism to NO which causes vasodilation and the relaxation of smooth muscle cells. The c...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Conditions:

Dexivacaine is a local anesthetic drug that has minimal and non-significant side effects.
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (ABSOLUTE)



Bepridil (trade name Vascor) is an amine calcium channel blocker used to treat angina. Bepridil is a calcium channel blocker that has well characterized anti-anginal properties and known but poorly characterized type 1 anti-arrhythmic and anti-hypert...
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (ACHIRAL)

Targets:

Azimilide is a class III antiarrhythmic agent that prolongs cardiac repolarisation by blocking both the rapidly and slowly activating components of the delayed rectifier potassium channel. The most important consequence of this is apparent rate-indep...
Status:
US Approved Rx (2024)
First approved in 1988

Class (Stereo):
CHEMICAL (RACEMIC)



Nicardipine is a potent calcium channel blockader with marked vasodilator action used to treat high blood pressure and angina. By deforming the channel, inhibiting ion-control gating mechanisms, and/or interfering with the release of calcium from the...
Status:
US Approved Rx (2017)
First approved in 1982

Class (Stereo):
CHEMICAL (ACHIRAL)



Piroxicam is in a class of drugs called nonsteroidal anti-inflammatory drugs (NSAIDs). It was originally brought to market by Pfizer under the tradename Feldene in 1980, became generic in 1992, and is marketed worldwide under many brandnames. Piroxic...