Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 22:16:22 GMT 2025
by
admin
on
Tue Apr 01 22:16:22 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
X6OG5T1C4M
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Q99720
Created by
admin on Tue Apr 01 22:16:22 GMT 2025 , Edited by admin on Tue Apr 01 22:16:22 GMT 2025
|
PRIMARY | |||
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X6OG5T1C4M
Created by
admin on Tue Apr 01 22:16:22 GMT 2025 , Edited by admin on Tue Apr 01 22:16:22 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
AGONIST -> TARGET |
Ki
|
||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Selective ligand of sigma sites in brain, labelled with (+)-[3 H] 3PPP (K i= 5.3±0.3 nM), were
investigated in rodents.
IC50
|
||
|
AGONIST -> TARGET | |||
|
AGONIST -> TARGET | |||
|
RADIOLIGAND->TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
AGONIST -> TARGET |
(+)-pentazocine is active
|
||
|
|
INHIBITOR -> TARGET |
Ki
|
||
|
AGONIST -> TARGET |
Ki
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
RADIOLIGAND->TARGET | |||
|
AGONIST -> TARGET |
IC50
|
||
|
AGONIST -> TARGET |
|
||
|
RADIOLIGAND->TARGET |
>146,000-fold selectivity over the ?2R and >10,000-fold selectivity over 59 different targets
Ki
|
||
|
INHIBITOR -> TARGET |
|
||
|
AGONIST -> TARGET |
Ki
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|