Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Sun Dec 18 14:00:13 UTC 2022
by
admin
on
Sun Dec 18 14:00:13 UTC 2022
|
Protein Type | RECEPTOR |
Protein Sub Type | |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
X6OG5T1C4M
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
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Common Name | English |
Code System | Code | Type | Description | ||
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Q99720
Created by
admin on Sun Dec 18 14:00:14 UTC 2022 , Edited by admin on Sun Dec 18 14:00:14 UTC 2022
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PRIMARY | |||
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X6OG5T1C4M
Created by
admin on Sun Dec 18 14:00:14 UTC 2022 , Edited by admin on Sun Dec 18 14:00:14 UTC 2022
|
PRIMARY |
Related Record | Type | Details | ||
---|---|---|---|---|
|
AGONIST -> TARGET |
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|
AGONIST -> TARGET | |||
|
AGONIST -> TARGET | |||
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RADIOLIGAND->TARGET |
IC50
|
||
|
AGONIST -> TARGET |
(+)-pentazocine is active
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INHIBITOR -> TARGET |
Ki
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INHIBITOR -> TARGET |
Ki
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||
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RADIOLIGAND->TARGET | |||
|
AGONIST -> TARGET |
IC50
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||
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RADIOLIGAND->TARGET |
>146,000-fold selectivity over the ?2R and >10,000-fold selectivity over 59 different targets
Ki
|
||
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AGONIST -> TARGET |
Ki
|
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|