U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sun Dec 18 08:03:23 UTC 2022
Edited
by admin
on Sun Dec 18 08:03:23 UTC 2022
Protein Type RECEPTOR
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
UKK18ES9TF
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
5-HYDROXYTRYPTAMINE RECEPTOR 1A
Common Name English
ADRB2RL1
Common Name English
5-HT1A
Common Name English
ADRBRL1
Common Name English
G-21
Common Name English
SEROTONIN RECEPTOR 1A
Common Name English
Code System Code Type Description
UNIPROT
P08908
Created by admin on Sun Dec 18 08:03:27 UTC 2022 , Edited by admin on Sun Dec 18 08:03:27 UTC 2022
PRIMARY
PHAROS
P08908
Created by admin on Sun Dec 18 08:03:27 UTC 2022 , Edited by admin on Sun Dec 18 08:03:27 UTC 2022
PRIMARY
FDA UNII
UKK18ES9TF
Created by admin on Sun Dec 18 08:03:27 UTC 2022 , Edited by admin on Sun Dec 18 08:03:27 UTC 2022
PRIMARY
From To
1_109 1_187
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_10
N 1_11
N 1_24
Related Record Type Details
AGONIST -> TARGET
INHIBITOR -> TARGET
PARTIAL AGONIST->TARGET
Ki
WEAK INHIBITOR->TARGET
INHIBITOR
Ki
RADIOLIGAND->TARGET
Kd
PARTIAL AGONIST->TARGET
Ki
INHIBITOR -> TARGET
AGONIST -> TARGET
PARTIAL AGONIST->TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST
Ki
AGONIST -> TARGET
AGONIST -> TARGET
RADIOLIGAND->TARGET
ACTIVATOR -> TARGET
INHIBITOR -> TARGET
Exhibited antagonism activity at both presynaptic and postsynaptic 5-HT1A receptor sites.
Kd
PARTIAL AGONIST->TARGET
Kd
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
LIGAND->TARGET
PARTIAL AGONIST->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
The strongest receptor binding affinity for 5-MeO-DiPT is at the 5-HT1A receptor.
AGONIST -> TARGET
SELECTIVE
PARTIAL AGONIST->TARGET
PARTIAL AGONIST->TARGET
Ki
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
Eletriptan binds with high affinity to 5-HT1B, 5-HT1D and 5-HT1F receptors, has modest affinity for 5-HT1A, 5-HT1E, 5-HT2B and 5-HT7 receptors
BINDING
PARTIAL AGONIST->TARGET
RADIOLIGAND->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
RADIOLIGAND->TARGET
Kd
RADIOLIGAND->TARGET
PARTIAL AGONIST->TARGET
INHIBITOR -> TARGET
INHIBITOR
Ki
AGONIST -> TARGET
AGONIST -> TARGET
RADIOLIGAND->TARGET
Kd
RADIOLIGAND->TARGET
Kd
RADIOLIGAND->TARGET
AGONIST -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL