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Showing 1 - 10 of 131 results

Status:
US Approved Rx (1983)
First approved in 1962

Class (Stereo):
CHEMICAL (RACEMIC)


Conditions:

Thioridazine (Mellaril or Melleril) is a piperidine typical antipsychotic drug belonging to the phenothiazine drug group and was previously widely used in the treatment of schizophrenia and psychosis. Thioridazine blocks postsynaptic mesolimbic dopam...
Status:
US Approved Rx (2016)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Glutodine (Cyproheptadine), sold under the brand name Periactin or Peritol, is a first-generation antihistamine with additional antiserotonergic, anticholinergic and local anesthetic properties. Glutodine is a white to slightly yellowish crystalline ...
Status:
US Approved Rx (1996)
First approved in 1959

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Fluphenazine is a trifluoro-methyl phenothiazine derivative intended for the management of schizophrenia and other psychotic disorders. Fluphenazine has not been shown effective in the management of behaviorial complications in patients with mental r...
Status:
US Approved Rx (2019)
First approved in 1946

Class (Stereo):
CHEMICAL (ABSOLUTE)



Methylergometrine (other names include methylergonovine, methylergobasin, methergine, and D-lysergic acid 1-butanolamide) is a synthetic analogue of ergonovine, a psychedelic alkaloid found in ergot, and many species of morning glory. In general, th...
Status:
US Approved Rx (2018)
First approved in 1946

Class (Stereo):
CHEMICAL (ABSOLUTE)


Conditions:

Dihydroergotamine (DHE) is a semisynthetic, hydrogenated ergot alkaloid, synthesized by reducing an unsaturated bond in ergotamine. Dihydroergotamine was originally envisaged as an antihypertensive agent, but it was later shown to be highly effective...
Status:
US Approved OTC
First approved in 2003

Class (Stereo):
CHEMICAL (ACHIRAL)



A sulfide ion is composed of a lone sulfur atom. Its charge is negative two, giving sulfides this formula: S^2-. Sulfide is a strong base, so solutions of sulfide in water are basic, due to hydrolysis. One well-known ionic compound with a sulfide ion...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Nelotanserin is a potent, selective 5-HT(2A) inverse agonist. Originally called ADP-125, the compound was developed by Arena Pharmaceuticals as a treatment for insomnia, but failed efficacy measures for this indication in Phase 2. In 2015, Axovant Sc...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)



Tiospirone (TSP) is an atypical antipsychotic drug. Tiaspirone appeared to be a promising antipsychotic agent as it didn`t cause extrapyramidal syndromes. It has 5HT-2 antagonistic properties as well as affinity for D2, 5HT-1a, 5HT-6 and sigma recep...
Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)


Metitepine, a psychotropic agent was developed as a non-selective antagonist of serotonin, dopamine, and adrenergic receptors. Metitepine has never been marketed.
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

m-Chlorophenylpiperazine (meta-chlorophenylpiperazine or mCPP) is a psychoactive substance, which is illegal in many countries but can be found on the black market. It induces endocrine, neurological and psychiatric effects. mCPP is a partial agonist...