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Showing 1 - 10 of 46 results

Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2022)
First approved in 1955

Class (Stereo):
CHEMICAL (ABSOLUTE)



Prednisolone is a synthetic adrenocortical steroid drug with predominantly glucocorticoid properties. Some of these properties reproduce the physiological actions of endogenous glucocorticosteroids, but others do not necessarily reflect any of the ad...
Status:
US Approved Rx (2003)
First approved in 1953

Class (Stereo):
CHEMICAL (RACEMIC)



Carbinoxamine is a histamine-H1 receptor blocking agent. It is an antihistamine with anticholinergic (drying) and sedative properties. Carbinoxamine appears to compete with histamine (type H1) for receptor sites on effector cells in the gastrointesti...
Status:
US Approved OTC
First marketed in 1901

Class (Stereo):
CHEMICAL (ABSOLUTE)



Epinephrine is a sympathomimetic catecholamine. It acts as a naturally occurring agonist at both alpha and beta-adrenergic receptors. Three pharmacologic types have been identified: alpha 1-, alpha 2-, and beta-adrenergic receptors. Each of these has...
Status:
US Animal Drug

Class (Stereo):
CHEMICAL (ABSOLUTE)

Conditions:

Flumethasone 21-acetate is an anti-inflammatory corticosteroid. It has 300 times greater anti-inflammatory activity and 677 times greater capacity to promote liver glycogen deposition than hydrocortisone. It has anti-rheumatic potency 31 times higher...
RS25344 is a potent and selective phosphodiesterase (PDE) 4 inhibitor. It preferentially inhibits phosphorylated PDE4D. The compound demonstrated efficacy in animal models of inflammation and anaphylaxis. RS25344 inhibited eosinophil chemotaxis, inc...
Status:
Other

Class (Stereo):
CHEMICAL (ACHIRAL)



ICI-63197 is a potent and selective phosphodiesterase IV (PDE 4) inhibitor with potent antidepressant activity. The antidepressant action of ICI-63197 realizes via enhancement of central noradrenergic transmission due to selective inhibition of cAMP ...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...