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Showing 1 - 10 of 16 results

Status:
US Approved Rx (2016)
First approved in 2002

Class (Stereo):
CHEMICAL (ABSOLUTE)



Voriconazole (vor-i-KON-a-zole, brand name Vfend, Pfizer) is a triazole antifungal medication. VFEND® (voriconazole) is available as film-coated tablets for oral administration, and as a lyophilized powder for solution for intravenous infusion. Vori...
Status:
US Approved Rx (2016)
First approved in 1992

Class (Stereo):
CHEMICAL (MIXED)



SPORANOX is the brand name for itraconazole, an azole antifungal agent. Itraconazole is a 1:1:1:1 racemic mixture of four diastereomers (two enantiomeric pairs), each possessing three chiral centers. In vitro studies have demonstrated that itraconazo...
Status:
US Approved Rx (2007)
First approved in 1992

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Terbinafine (brand name Lamisil, Terbisil, Terboderm and others) is an antifungal medication used to treat ringworm and fungal nail infections. Terbinafine inhibits ergosterol synthesis by inhibiting squalene epoxidase, an enzyme that is part of the...
Status:
US Approved Rx (2005)
First approved in 1987

Class (Stereo):
CHEMICAL (RACEMIC)



Terconazole is an antifungal drug used to treat vaginal yeast infection. Terconazole may exert its antifungal activity by disrupting normal fungal cell membrane permeability. Terconazole and other triazole antifungal agents inhibit cytochrome P450 "1...
Status:
US Approved Rx (2007)
First approved in 1959

Class (Stereo):
CHEMICAL (ABSOLUTE)



Griseofulvin is a mycotoxic metabolic product of Penicillium spp. It was the first available oral agent for the treatment of dermatophytoses and has now been used for more than forty years. Griseofulvin is fungistatic with in vitro activity against v...
Status:
Possibly Marketed Outside US
First approved in 2000

Class (Stereo):
CHEMICAL (ACHIRAL)

Conditions:

Isopropyl Myristate is a synthetic oil used as an emollient, thickening agent or lubricant in beauty products. Isopropyl Myristate is a popular cosmetic and pharmaceutical ingredient. It is most often used as an additive in aftershaves, shampoos, bat...
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (RACEMIC)


Conditions:

Enilconazole is a synthetic broad-spectrum antimycotic with a high activity against most of the common dermatophytes and various other fungi and yeasts. It is a selective inhibitor of ergosterol biosynthesis, an essential component of the cell membra...
Status:
US Approved Rx (2016)
First approved in 2002

Class (Stereo):
CHEMICAL (ABSOLUTE)



Voriconazole (vor-i-KON-a-zole, brand name Vfend, Pfizer) is a triazole antifungal medication. VFEND® (voriconazole) is available as film-coated tablets for oral administration, and as a lyophilized powder for solution for intravenous infusion. Vori...
Status:
US Approved Rx (2016)
First approved in 2002

Class (Stereo):
CHEMICAL (RACEMIC)



Voriconazole (vor-i-KON-a-zole, brand name Vfend, Pfizer) is a triazole antifungal medication. VFEND® (voriconazole) is available as film-coated tablets for oral administration, and as a lyophilized powder for solution for intravenous infusion. Vori...

Showing 1 - 10 of 16 results