U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sun Dec 18 09:15:51 UTC 2022
Edited
by admin
on Sun Dec 18 09:15:51 UTC 2022
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
EV0PWK6TT6
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
DELTA-TYPE OPIOID RECEPTOR
Common Name English
OPRD
Common Name English
Code System Code Type Description
PHAROS
P41143
Created by admin on Sun Dec 18 09:15:53 UTC 2022 , Edited by admin on Sun Dec 18 09:15:53 UTC 2022
PRIMARY
FDA UNII
EV0PWK6TT6
Created by admin on Sun Dec 18 09:15:53 UTC 2022 , Edited by admin on Sun Dec 18 09:15:53 UTC 2022
PRIMARY
UNIPROT
P41143
Created by admin on Sun Dec 18 09:15:53 UTC 2022 , Edited by admin on Sun Dec 18 09:15:53 UTC 2022
PRIMARY
From To
1_121 1_198
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_18
N 1_33
Related Record Type Details
PARTIAL AGONIST->TARGET
EMAX = 28% OF DAMGO
EC50
AGONIST -> TARGET
AGONIST -> TARGET
SELECTIVE
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
ANTAGONIST
RADIOLIGAND->TARGET
PARENT->INNOVATOR
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
SELECTIVE FOR DELTA AND DELTA-MU heteromers[
INHIBITOR -> TARGET
INHIBITOR -> TARGET
PARTIAL AGONIST->TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
WEAK AGONIST->TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
In the MVD, C8813 could inhibit the electrically induced contraction, but weaker than in the GPI. Moreover, this inhibitory effect could antagonized by the ?-opioid receptor antagonist ICI174864. These results indicated C8813 also acted on ?-opioid receptor but less potent than on ?-opioid receptor.
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL