Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 21:20:47 GMT 2025
by
admin
on
Tue Apr 01 21:20:47 GMT 2025
|
| Protein Type | SIGNAL TRANSDUCER |
| Protein Sub Type | TRANSCRIPTION ACTIVATOR |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
51F8I2CLT3
|
| Record Status |
Validated (UNII)
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| Record Version |
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-
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| Name | Type | Language | ||
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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51F8I2CLT3
Created by
admin on Tue Apr 01 21:20:47 GMT 2025 , Edited by admin on Tue Apr 01 21:20:47 GMT 2025
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PRIMARY | |||
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P40763
Created by
admin on Tue Apr 01 21:20:47 GMT 2025 , Edited by admin on Tue Apr 01 21:20:47 GMT 2025
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PRIMARY |
| Related Record | Type | Details | ||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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ACTIVATOR -> TARGET |
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INHIBITOR -> TARGET |
In HepG2 cells, in the presence of 50 pM IL-6 (luciferase assay)
INHIBITOR
IC50
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INHIBITOR OF EXPRESSION->TARGET | |||
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INHIBITOR -> TARGET |
Inhibits phosphorylation, cell proliferation and induces apoptosis.
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INDUCER -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR OF EXPRESSION->TARGET | |||
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INHIBITOR -> TARGET |
Inhibits the activation of STAT3 signaling resulting from tyrosine residue phosphorylation (Y705) leads to aberrant oncogene transcription.
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
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