Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Fri Jun 25 21:36:10 UTC 2021
by
admin
on
Fri Jun 25 21:36:10 UTC 2021
|
Protein Type | RECEPTOR |
Protein Sub Type | KINASE |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
1L68U00N7O
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
Name | Type | Language | ||
---|---|---|---|---|
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
Code System | Code | Type | Description | ||
---|---|---|---|---|---|
|
1L68U00N7O
Created by
admin on Fri Jun 25 21:36:10 UTC 2021 , Edited by admin on Fri Jun 25 21:36:10 UTC 2021
|
PRIMARY | |||
|
P04629
Created by
admin on Fri Jun 25 21:36:10 UTC 2021 , Edited by admin on Fri Jun 25 21:36:10 UTC 2021
|
PRIMARY | |||
|
P04629
Created by
admin on Fri Jun 25 21:36:10 UTC 2021 , Edited by admin on Fri Jun 25 21:36:10 UTC 2021
|
PRIMARY |
From | To |
---|---|
1_122 | 1_159 |
1_183 | 1_233 |
Glycosylation Type | HUMAN |
Glycosylation Link Type | Site |
---|---|
N | 1_35 |
N | 1_63 |
N | 1_89 |
N | 1_156 |
N | 1_170 |
N | 1_221 |
N | 1_230 |
N | 1_249 |
N | 1_286 |
N | 1_291 |
N | 1_306 |
N | 1_326 |
N | 1_369 |
Related Record | Type | Details | ||
---|---|---|---|---|
|
INHIBITOR -> TARGET |
Active against NTRK gene fusions. Competitive to ATP binding site.
COMPETITIVE INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
AGONIST -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT | CHEMICAL |
|
||||
Molecular Formula | CHEMICAL |
|