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Showing 131 - 140 of 13,259 results

Status:
US Approved Rx (2017)
First approved in 1992

Class (Stereo):
CHEMICAL (ACHIRAL)



Oxaprozin is a nonsteroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Anti-inflammatory effects of Oxaprozin are believed to be due to inhibition of cylooxygenase in platelets which leads to the blockage of prostagland...
Status:
US Approved Rx (2021)
First approved in 1992

Class (Stereo):
CHEMICAL (ACHIRAL)



Sumatriptan is a serotonin (5-HT1B/1D) receptor agonist indicated for acute treatment of migraine with or without aura in adults. Sumatriptan is structurally similar to serotonin (5-HT), and is a 5-HT receptor (types 5-HT1D and 5-HT1B) agonist. The ...
Status:
US Approved Rx (1999)
First approved in 1992

Class (Stereo):
CHEMICAL (ABSOLUTE)


Conditions:

Desogestrel is a prodrug of etonogestrel (3-keto-desogestrel) which was approved as oral contraceptove medicine. Desogestrel acts selectively binding to progesterone receptor and enchancing its activity.
Status:
US Approved Rx (2007)
First approved in 1991

Class (Stereo):
CHEMICAL (ABSOLUTE)



Histrelin is a gonadotropin releasing hormone (GnRH) agonist that acts as a potent inhibitor of gonadotropin when administered as an implant that delivers continuous therapeutic doses. Following an initial stimulatory phase with increased circulating...
Status:
US Approved Rx (2010)
First approved in 1991

Class (Stereo):
CHEMICAL (RACEMIC)


Conditions:

Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker (CCB)b. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium...
Status:
US Approved Rx (2020)
First approved in 1991

Class (Stereo):
CHEMICAL (RACEMIC)



Etodolac is an anti-inflammatory agent with analgesic and antipyretic properties. It is used to treat osteoarthritis, rheumatoid arthritis and control acute pain. The therapeutic effects of etodolac are achieved via inhibition of the synthesis of pro...
Status:
US Approved Rx (2012)
First approved in 1991

Class (Stereo):
CHEMICAL (ACHIRAL)



Fumazenil is an imidazobenzodiazepine derivative and a potent benzodiazepine receptor antagonist that competitively inhibits the activity at the benzodiazepine recognition site on the GABA/benzodiazepine receptor complex, thereby reversing the effect...
Status:
US Approved Rx (2007)
First approved in 1991

Class (Stereo):
CHEMICAL (ABSOLUTE)


Conditions:

Prednicarbate is a relatively new topical corticosteroid drug. It is similar in potency to hydrocortisone. It has a favorable benefit-risk ratio, with an inflammatory action similar to that of a medium potency corticosteroid, but with a low potential...
Status:
US Approved Rx (1997)
First approved in 1990

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Estazolam, a triazolobenzodiazepine derivative, is an oral hypnotic agent with anticonvulsant, hypnotic, and muscle relaxant properties. It has been shown in some cases to be more potent than diazepam or nitrazepam. Benzodiazepines bind nonspecifical...
Status:
US Approved Rx (2024)
First approved in 1988

Class (Stereo):
CHEMICAL (RACEMIC)



Nicardipine is a potent calcium channel blockader with marked vasodilator action used to treat high blood pressure and angina. By deforming the channel, inhibiting ion-control gating mechanisms, and/or interfering with the release of calcium from the...

Showing 131 - 140 of 13,259 results