U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}

    {{facet.count}}
    {{facet.count}}
Status:
Investigational
Source:
INN:myfadol
Source URL:

Class (Stereo):
CHEMICAL (MIXED)

Myfadol is a phenacylpiperidine derivative patented by Tanabe Seiyaku Co., Ltd as low molecular weight non-peptide analgesic. Myfadol produces hot-plate analgesia in rodents with minimal side-effects, and when given parenterally in humans produces analgesia to experimentally-produced and postoperative pain.
Status:
Investigational
Source:
INN:felipyrine [INN]
Source URL:

Class (Stereo):
CHEMICAL (RACEMIC)


Felipyrine is a 1-aryl-2-pyrrolidinone derivative exerting anti-inflammatory activity.
Status:
Investigational
Source:
INN:quatacaine
Source URL:

Class (Stereo):
CHEMICAL (ACHIRAL)

Quatacaine is a methylpropionanilide derivative patented by Tanabe Seiyaku Co., Ltd. As local anaesthetic.
Status:
Investigational
Source:
INN:tiapirinol [INN]
Source URL:

Class (Stereo):
CHEMICAL (MIXED)

Tiapirinol is a thiazine derivative patented by Tanabe Seiyaku Co., Ltd. as a low toxic compound useful to prevent hypohepatia. In acute toxicity tests on mice, the toxicity of Tiapirinol is lower than that of pyridoxal phosphate and other vitamin B6 derivative. Tiapirinol showed vitamin B6 activity approximately equivalent to that of pyridoxal phosphate or pyridoxine for the growth of vitamin B6 deficient rats and also for the convulsions caused by antivitamin B6 agents.
Status:
Investigational
Source:
JAN:MAFOPRAZINE MESILATE [JAN]
Source URL:

Class (Stereo):
CHEMICAL (ACHIRAL)


Mafoprazine is a phenylpiperazine derivative exerting postsynaptic dopamine D2 receptor blocking activity and alpha-adrenergic activity (alpha 1 receptor blocking activity and alpha 2 receptor stimulating activity). In animal models, mafoprazine demonstrated antipsychotic, aggression-inhibiting and cataleptogenic actions.
Status:
Investigational
Source:
JAN:MAFOPRAZINE MESILATE [JAN]
Source URL:

Class (Stereo):
CHEMICAL (ACHIRAL)


Mafoprazine is a phenylpiperazine derivative exerting postsynaptic dopamine D2 receptor blocking activity and alpha-adrenergic activity (alpha 1 receptor blocking activity and alpha 2 receptor stimulating activity). In animal models, mafoprazine demonstrated antipsychotic, aggression-inhibiting and cataleptogenic actions.
Status:
Investigational
Source:
INN:myfadol
Source URL:

Class (Stereo):
CHEMICAL (MIXED)

Myfadol is a phenacylpiperidine derivative patented by Tanabe Seiyaku Co., Ltd as low molecular weight non-peptide analgesic. Myfadol produces hot-plate analgesia in rodents with minimal side-effects, and when given parenterally in humans produces analgesia to experimentally-produced and postoperative pain.
Status:
Investigational
Source:
INN:quatacaine
Source URL:

Class (Stereo):
CHEMICAL (ACHIRAL)

Quatacaine is a methylpropionanilide derivative patented by Tanabe Seiyaku Co., Ltd. As local anaesthetic.
Status:
Investigational
Source:
INN:myfadol
Source URL:

Class (Stereo):
CHEMICAL (MIXED)

Myfadol is a phenacylpiperidine derivative patented by Tanabe Seiyaku Co., Ltd as low molecular weight non-peptide analgesic. Myfadol produces hot-plate analgesia in rodents with minimal side-effects, and when given parenterally in humans produces analgesia to experimentally-produced and postoperative pain.