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Showing 1 - 10 of 53 results

Status:
US Approved Rx (2018)
First approved in 2018

Class (Stereo):
CHEMICAL (ACHIRAL)



Prucalopride is a novel enterokinetic compound and is the first representative of the benzofuran class. Prucalopride is a potent, selective and specific serotonin 5-HT4 receptor (5-HT4-R) agonist. Prucalopride (Resolor®), a highly selective serotonin...
Status:
US Approved Rx (1999)
First approved in 1986

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Alfentanil is an opioid analgesic with a rapid onset of action. Alfentanil interacts predominately with the opioid mu-receptor. These mu-binding sites are discretely distributed in the human brain, spinal cord, and other tissues. In clinical settings...
Status:
US Approved Rx (2004)
First approved in 1970

Class (Stereo):
CHEMICAL (ACHIRAL)



Flavoxate is a drug, indicated for symptomatic relief of dysuria, urgency, nocturia, suprapubic pain, frequency and incontinence as may occur in cystitis, prostatitis, urethritis, urethrocystitis/urethrotrigonitis. Flavoxate is not indicated for defi...
Status:
US Approved Rx (1968)
First approved in 1968

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Fentanyl is a potent agonist of mu opioid receptor. It is used to relieve severe pain, such as after surgery or during cancer treatment, and breakthrough pain (flare-ups of intense pain despite round-the-clock narcotic treatment). Fentanyl is an extr...
Status:
US Approved Rx (1988)
First approved in 1968

Class (Stereo):
CHEMICAL (RACEMIC)



Droperidol produces marked tranquilization and sedation. It allays apprehension and provides a state of mental detachment and indifference while maintaining a state of reflex alertness. Droperidol produces an antiemetic effect as evidenced by the ant...
Status:
US Approved Rx (2007)
First approved in 1967

Class (Stereo):
CHEMICAL (ACHIRAL)



Haloperidol is a phenyl-piperidinyl-butyrophenone that is used primarily to treat schizophrenia and other psychoses. It is also used in schizoaffective disorder, delusional disorders, ballism, and Tourette syndrome (a drug of choice) and occasionally...
Status:
US Approved OTC
First approved in 1974

Class (Stereo):
CHEMICAL (RACEMIC)



Miconazole is a synthetic imidazole derivative, a topical antifungal agent for use in the local treatment of vaginal, and skin and nail infections due to yeasts and dermatophytes. It is particularly active against Candida spp., Trichophyton spp., Epi...
Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)


Meletimide (R 5183) is a powerful anticholinergic agent with pronounced peripheral and central action.
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Mavatrep (JNJ-39439335) is a TRPV1 antagonist. It exerts analgesic potential. Mavatrep demonstrated sustained pharmacodynamic effects (heat pain perception, heat pain latency, capsaicin-induced flare), and an efficacy signal in participants with oste...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Lusaperidone (R107474) is a potent and relatively selective alpha(2)-adrenoceptor antagonist. It was under clinical evaluation for the treatment of depression, characterized by anergia and lack of drive. However, further clinical development has been...