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Showing 1 - 10 of 21 results

Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2003)
First approved in 1953

Class (Stereo):
CHEMICAL (RACEMIC)



Carbinoxamine is a histamine-H1 receptor blocking agent. It is an antihistamine with anticholinergic (drying) and sedative properties. Carbinoxamine appears to compete with histamine (type H1) for receptor sites on effector cells in the gastrointesti...
Status:
US Previously Marketed
First approved in 1960

Class (Stereo):
CHEMICAL (ABSOLUTE)



Rotoxamine ((S)-carbinoxamine) is maleic acid salt of the levorotatory isomer of Carbinoxamine (a first-generation antihistamine of the ethanolamine class). Ethanolamine antihistamines have significant antimuscarinic activity and produce marked sedat...
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (ACHIRAL)



Mebhydrolin (INN) or mebhydroline is a histamine H1-receptor antagonist. It is not available in the United States, but it is available in various other countries under the brand names Bexidal and Diazolin. It is used for symptomatic relief of allergi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ABSOLUTE)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...
Status:
US Approved Rx (2006)
First approved in 1961

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyproheptadine hydrochloride anhydrous is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties. It is indicted for the treatment of perennial and seasonal allergic rhinitis; vasomotor rhi...