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Showing 1 - 10 of 76 results

Status:
US Approved Rx (1995)
First approved in 1977

Class (Stereo):
CHEMICAL (ACHIRAL)



Cyclobenzaprine is a centrally-acting muscle relaxant which boosts levels of norepinephrine and binds to serotonin receptors in the brain to reduce spasm. Cytochromes P-450 3A4, 1A2, and, to a lesser extent, 2D6, mediate N-demethylation, one of the o...
Status:
US Approved Rx (1985)
First approved in 1977

Class (Stereo):
CHEMICAL (RACEMIC)



Disopyramide is an antiarrhythmic drug indicated for the treatment of documented ventricular arrhythmias, such as sustained ventricular tachycardia that are life-threatening. In man, Disopyramide at therapeutic plasma levels shortens the sinus node r...
Status:
US Approved Rx (2024)
First approved in 1977

Class (Stereo):
CHEMICAL (ACHIRAL)



Cimetidine is a histamine H2-receptor antagonist. It reduces basal and nocturnal gastric acid secretion and a reduction in gastric volume, acidity, and amount of gastric acid released in response to stimuli including food, caffeine, insulin, betazole...
Status:
US Approved Rx (2003)
First approved in 1977

Class (Stereo):
CHEMICAL (ACHIRAL)



Tamoxifen (brand name Nolvadex), is selective estrogen receptor modulators (SERM) with tissue-specific activities for the treatment and prevention of estrogen receptor positive breast cancer. Tamoxifen itself is a prodrug, having relatively little af...
Status:
US Approved Rx (1979)
First approved in 1977

Class (Stereo):
CHEMICAL (ACHIRAL)


Thallous chloride (also known as Thallium(I) chloride) is a chemical compound with the formula TlCl. Thallous Chloride Tl 201 Injection is a diagnostic radiopharmaceutical indicated for: Myocardial perfusion imaging with planar scintigraphy or single...
Status:
US Approved Rx (2017)
First approved in 1977

Class (Stereo):
CHEMICAL (ABSOLUTE)



Diflorasone is a topical corticosteroid used to treat itching and inflammation of the skin. Topical corticosteroids share anti-inflammatory, antipruritic and vasoconstrictive actions. The mechanism of anti-inflammatory activity of the topical cortico...
Status:
US Approved Rx (1997)
First approved in 1977

Class (Stereo):
CHEMICAL (ABSOLUTE)



Clemastine is an antihistamine with anticholinergic (drying) and sedative side effects. Clemastine is a selective histamine H1 antagonist and binds to the histamine H1 receptor. This blocks the action of endogenous histamine, which subsequently leads...
Status:
US Approved Rx (2007)
First approved in 1977

Class (Stereo):
CHEMICAL (RACEMIC)


Conditions:

Baclofen (brand names Kemstro, Lioresal, and Gablofen) is a derivative of gamma-aminobutyric acid (GABA). Baclofen is a muscle relaxer and an antispastic agent and is used to treat muscle symptoms caused by multiple sclerosis, including spasm, pain, ...
Status:
US Approved Rx (2001)
First approved in 1977

Class (Stereo):
CHEMICAL (RACEMIC)


Conditions:

Lorazepam (brand name Ativan) is indicated for the management of anxiety disorders or for the short-term relief of the symptoms of anxiety or anxiety associated with depressive symptoms. Anxiety or tension associated with the stress of everyday life ...
Status:
US Approved Rx (1992)
First approved in 1977

Class (Stereo):
CHEMICAL (ABSOLUTE)



Dinoprostone is a naturally occurring prostaglandin E2 (PGE2). Dinoprostone is equivalent to prostaglandin E2 (PGE2). It stimulates labor and delivery by stimulating the uterine, and thus terminates pregnancy. Dinoprostone is also capable of stimulat...