Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:37:46 GMT 2025
by
admin
on
Tue Apr 01 18:37:46 GMT 2025
|
Protein Sub Type | |
Sequence Type | COMPLETE |
Record UNII |
XGE1085C9Q
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
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XGE1085C9Q
Created by
admin on Tue Apr 01 18:37:46 GMT 2025 , Edited by admin on Tue Apr 01 18:37:46 GMT 2025
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PRIMARY | |||
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P42338
Created by
admin on Tue Apr 01 18:37:46 GMT 2025 , Edited by admin on Tue Apr 01 18:37:46 GMT 2025
|
PRIMARY |
Related Record | Type | Details | ||
---|---|---|---|---|
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Ki
|
||
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WEAK INHIBITOR->TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
INHIBITOR
IC50
|
||
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INHIBITOR -> TARGET |
Ki
|
||
|
NON-INHIBITOR->OFF TARGET |
IC50
|
||
|
WEAK INHIBITOR->OFF TARGET |
IC50
|
||
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INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
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SUBSTRATE -> TARGET |
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INHIBITOR -> TARGET |
IC50
|
||
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INHIBITOR -> TARGET |
|
||
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INHIBITOR -> TARGET |
INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
WEAK INHIBITOR->OFF TARGET |
IC50
|
||
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WEAK INHIBITOR->OFF TARGET |
RLY-2608 shows potent isoform
selective, biochemical inhibition
IC50
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||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
HTRF technology assay.
IC50
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Structural Modifications
Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
---|---|---|---|---|---|---|
AMINO ACID SUBSTITUTION | [1_324] [1_1070] | S | TYROSINE O-PHOSPHATE | 2R86C98KDX |
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT | CHEMICAL |
|