AM-2201

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National Institutes of Health Divider Arrow

NCATS

Details

Stereochemistry	ACHIRAL
Molecular Formula	C24H22FNO
Molecular Weight	359.436
Optical Activity	NONE
Defined Stereocenters	0 / 0
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure of AM-2201

Structure Search

SMILES

FCCCCCN1C=C(C(=O)C2=CC=CC3=C2C=CC=C3)C4=C1C=CC=C4

InChI

InChIKey=ALQFAGFPQCBPED-UHFFFAOYSA-N

InChI=1S/C24H22FNO/c25-15-6-1-7-16-26-17-22(20-12-4-5-14-23(20)26)24(27)21-13-8-10-18-9-2-3-11-19(18)21/h2-5,8-14,17H,1,6-7,15-16H2

HIDE SMILES / InChI

Molecular Formula	C24H22FNO
Molecular Weight	359.436
Charge	0
Count

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Approval Year

Targets

Targets

Primary Target	Pharmacology	Condition	Potency
Cannabinoid CB1 receptor 85 Target ID: CHEMBL218 Sources: https://www.ncbi.nlm.nih.gov/pubmed/25921407 \| https://legal-high-inhaltsstoffe.de/sites/default/files/uploads/am-2201.pdf \| https://www.ncbi.nlm.nih.gov/pubmed/30280499	Agonist 2678		38.0 nM [EC50]
Cannabinoid CB2 receptor 71 Target ID: CHEMBL253 Sources: https://www.ncbi.nlm.nih.gov/pubmed/25921407	Agonist 2678		2.6 nM [Ki]

PubMed

PubMed

Title	Date	PubMed
Genotoxic properties of representatives of alkylindazoles and aminoalkyl-indoles which are consumed as synthetic cannabinoids.	2015 Jun	25792264

Substance Class	Chemical Created by `admin` on `Sat Dec 16 07:15:39 UTC 2023` Edited by `admin` on `Sat Dec 16 07:15:39 UTC 2023`
Record UNII	TBJ0966F1O
Record Status	`Validated (UNII)`
Record Version

Download

Name

Type

Language

AM-2201

Common Name

English

1-(5-FLUOROPENTYL)-3-(1-NAPHTHOYL)INDOLE

Systematic Name

English

JWH-2201

Code

English

AM2201

Code

English

METHANONE, (1-(5-FLUOROPENTYL)-1H-INDOL-3-YL)-1-NAPHTHALENYL-

Systematic Name

English

DEA NO. 7201

Code

English

J2.973.653G

Code

English

Classification Tree Code System Code

DEA NO.

7201

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

WIKIPEDIA

Designer-drugs-AM-2201

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

Code System Code Type Description

CAS

335161-24-5

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

PRIMARY

EPA CompTox

DTXSID50187158

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

PRIMARY

SMS_ID

100000183990

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

PRIMARY

WIKIPEDIA

AM-2201

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

PRIMARY

FDA UNII

TBJ0966F1O

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

PRIMARY

PUBCHEM

53393997

Created by admin on Sat Dec 16 07:15:39 UTC 2023 , Edited by admin on Sat Dec 16 07:15:39 UTC 2023

PRIMARY

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TARGET -> AGONIST

Comments:

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Qualification:

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					TBJ0966F1O

AM-2201

ACTIVE MOIETY