Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Mon Mar 31 20:36:53 GMT 2025
by
admin
on
Mon Mar 31 20:36:53 GMT 2025
|
| Protein Type | GROWTH FACTOR |
| Protein Sub Type | TGF .BETA. SUPERFAMILY |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
T7D25J14LT
|
| Record Status |
Validated (UNII)
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| Record Version |
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-
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| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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T7D25J14LT
Created by
admin on Mon Mar 31 20:36:53 GMT 2025 , Edited by admin on Mon Mar 31 20:36:53 GMT 2025
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PRIMARY | |||
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P01137
Created by
admin on Mon Mar 31 20:36:53 GMT 2025 , Edited by admin on Mon Mar 31 20:36:53 GMT 2025
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PRIMARY | |||
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T7D25J14LT
Created by
admin on Mon Mar 31 20:36:53 GMT 2025 , Edited by admin on Mon Mar 31 20:36:53 GMT 2025
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PRIMARY | |||
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C1293
Created by
admin on Mon Mar 31 20:36:53 GMT 2025 , Edited by admin on Mon Mar 31 20:36:53 GMT 2025
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PRIMARY | |||
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1426465
Created by
admin on Mon Mar 31 20:36:53 GMT 2025 , Edited by admin on Mon Mar 31 20:36:53 GMT 2025
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PRIMARY | |||
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300000025998
Created by
admin on Mon Mar 31 20:36:53 GMT 2025 , Edited by admin on Mon Mar 31 20:36:53 GMT 2025
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PRIMARY |
| From | To |
|---|---|
| 1_7 | 1_16 |
| 1_15 | 1_78 |
| 1_44 | 1_109 |
| 1_48 | 1_111 |
| 1_77 | 2_77 |
| 2_7 | 2_16 |
| 2_15 | 2_78 |
| 2_44 | 2_109 |
| 2_48 | 2_111 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
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LIGAND->TARGET |
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INHIBITOR -> TARGET |
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VECTOR->EXPRESSED PROTEIN |
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INHIBITOR OF EXPRESSION->TARGET |
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INHIBITOR -> TARGET |
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TARGET -> AGONIST |
TGFB1, TGFB2 and TGFB3 homodimeric ligands assemble a functional receptor composed of two TGFBR1 and TGFBR2 heterodimers to form a ligand-receptor heterohexamer.
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TARGE->INHIBITION OF ACTIVATION |
Inhibited Smad2 phosphorylation in a concentration-dependent manner
EC50
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INHIBITOR -> TARGET |
IN-VITRO
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INHIBITOR OF EXPRESSION->TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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| Related Record | Type | Details | ||
|---|---|---|---|---|
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ACTIVE MOIETY |
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
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| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
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