U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 13:58:55 UTC 2023
Edited
by admin
on Sat Dec 16 13:58:55 UTC 2023
Protein Type ENZYME
Protein Sub Type KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
T59477XR5I
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TYROSINE-PROTEIN KINASE BTK C481S (IBRUTINIB RESISTANT MUTANT)
Common Name English
BTK C481S
Common Name English
TYROSINE-PROTEIN KINASE BTK C481S MUTANT (METHIONINE INCLUDED IN NUMBERING)
Common Name English
TYROSINE-PROTEIN KINASE BTK C480S MUTANT
Common Name English
Code System Code Type Description
FDA UNII
T59477XR5I
Created by admin on Sat Dec 16 13:58:56 UTC 2023 , Edited by admin on Sat Dec 16 13:58:56 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
REVERSIBLE
IC50
INHIBITOR -> TARGET
IN-VITRO
INHIBITOR -> TARGET
IC50
INHIBITOR RESISTANT -> TARGET
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL