OLICERIDINE

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National Institutes of Health Divider Arrow

NCATS

Details

Stereochemistry	ABSOLUTE
Molecular Formula	C22H30N2O2S
Molecular Weight	386.551
Optical Activity	UNSPECIFIED
Defined Stereocenters	1 / 1
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure of OLICERIDINE

Structure Search

SMILES

COC1=C(CNCC[C@]2(CCOC3(CCCC3)C2)C4=NC=CC=C4)SC=C1

InChI

InChIKey=DMNOVGJWPASQDL-OAQYLSRUSA-N

InChI=1S/C22H30N2O2S/c1-25-18-7-15-27-19(18)16-23-13-10-21(20-6-2-5-12-24-20)11-14-26-22(17-21)8-3-4-9-22/h2,5-7,12,15,23H,3-4,8-11,13-14,16-17H2,1H3/t21-/m1/s1

HIDE SMILES / InChI

Molecular Formula	C22H30N2O2S
Molecular Weight	386.551
Charge	0
Count

Stereochemistry	ABSOLUTE
Additional Stereochemistry	No
Defined Stereocenters	1 / 1
E/Z Centers	0
Optical Activity	UNSPECIFIED

Approval Year

Substance Class	Chemical Created by `admin` on `Sun Dec 18 17:52:02 UTC 2022` Edited by `admin` on `Sun Dec 18 17:52:02 UTC 2022`
Record UNII	MCN858TCP0
Record Status	`Validated (UNII)`
Record Version

Download

Name

Type

Language

OLICERIDINE

Official Name

English

Oliceridine [WHO-DD]

Common Name

English

TRV130

Code

English

oliceridine [INN]

Common Name

English

TRV-130

Code

English

OLICERIDINE [MI]

Common Name

English

6-OXASPIRO(4.5)DECANE-9-ETHANAMINE, N-((3-METHOXY-2-THIENYL)METHYL)-9-(2-PYRIDINYL)-, (9R)-

Systematic Name

English

OLICERIDINE [ORANGE BOOK]

Common Name

English

OLICERIDINE [USAN]

Common Name

English

N-[(3-Methoxythiophen-2-yl)methyl]-2-[(9R)-9-(pyridin-2-yl)-6-oxaspiro[4.5]decan-9-yl]ethanamine

Systematic Name

English

OLINVYK

Brand Name

English

Classification Tree Code System Code

DEA NO.

9245

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

Code System Code Type Description

CAS

1401028-24-7

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

DRUG BANK

DB14881

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

INN

10250

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

NCI_THESAURUS

C174704

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

MERCK INDEX

M12219

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

WIKIPEDIA

Oliceridine

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

PUBCHEM

66553195

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

EPA CompTox

DTXSID201031292

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

FDA UNII

MCN858TCP0

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

USAN

CD-26

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

RXCUI

2392230

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

ChEMBL

CHEMBL2443262

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

DAILYMED

MCN858TCP0

Created by admin on Sun Dec 18 17:52:03 UTC 2022 , Edited by admin on Sun Dec 18 17:52:03 UTC 2022

PRIMARY

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ACTIVE MOIETY

Name	Property Type	Amount	Referenced Substance	Defining	Parameters	References
Volume of Distribution	PHARMACOKINETIC				AT STEADY-STATE

Tmax	PHARMACOKINETIC				SINGLE DOSE INTRAVENOUS ADMINISTRATION

Biological Half-life	PHARMACOKINETIC				INTRAVENOUS ADMINISTRATION SINGLE DOSE