Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 17:39:47 GMT 2025
by
admin
on
Tue Apr 01 17:39:47 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
M4PJ7V12VY
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Q16620
Created by
admin on Tue Apr 01 17:39:48 GMT 2025 , Edited by admin on Tue Apr 01 17:39:48 GMT 2025
|
PRIMARY | |||
|
M4PJ7V12VY
Created by
admin on Tue Apr 01 17:39:48 GMT 2025 , Edited by admin on Tue Apr 01 17:39:48 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_1 | 1_7 |
| 1_5 | 1_14 |
| 1_121 | 1_145 |
| 1_123 | 1_163 |
| 1_187 | 1_235 |
| 1_271 | 1_314 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_36 |
| N | 1_64 |
| N | 1_90 |
| N | 1_147 |
| N | 1_174 |
| N | 1_210 |
| N | 1_223 |
| N | 1_249 |
| N | 1_294 |
| N | 1_307 |
| N | 1_381 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
ANTAGONIST
|
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|
PARTIAL AGONIST->TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
COMPETITIVE INHIBITOR
IC50
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||
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|
INHIBITOR -> TARGET |
|
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|
INHIBITOR -> TARGET |
IC50
|
||
|
AGONIST -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR->OFF-TARGET |
|
||
|
RADIOLIGAND->TARGET |
Through a panel of 369 human kinases (no detectable kinase off-target at 1000-fold concentration over TrkB/C potency)
IC50
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET | |||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
|
||
|
AGONIST -> TARGET | |||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
AGONIST -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_485] [1_671] [1_675] [1_676] [1_786] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|