U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 09:11:38 UTC 2023
Edited
by admin
on Sat Dec 16 09:11:38 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
G49RZO51ZC
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
OATP-B
Common Name English
SLC21A9
Common Name English
SLCO2B1
Common Name English
OATP2B1
Common Name English
ORGANIC ANION TRANSPORTER POLYPEPTIDE-RELATED PROTEIN 2
Common Name English
DKFZP686E0517
Common Name English
SOLUTE CARRIER ORGANIC ANION TRANSPORTER FAMILY MEMBER 2B1
Common Name English
KIAA0880
Common Name English
OATPB
Common Name English
OATPRP2
Common Name English
Classification Tree Code System Code
UCSF-FDA TRANSPORTAL SLCO2B1
Created by admin on Sat Dec 16 09:11:39 UTC 2023 , Edited by admin on Sat Dec 16 09:11:39 UTC 2023
Code System Code Type Description
UNIPROT
Q9Y6L6
Created by admin on Sat Dec 16 09:11:39 UTC 2023 , Edited by admin on Sat Dec 16 09:11:39 UTC 2023
PRIMARY
FDA UNII
G49RZO51ZC
Created by admin on Sat Dec 16 09:11:39 UTC 2023 , Edited by admin on Sat Dec 16 09:11:39 UTC 2023
PRIMARY
From To
1_489 1_516
1_493 1_504
1_495 1_520
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_176
N 1_538
Related Record Type Details
INHIBITOR -> TRANSPORTER
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: ESTRONE-3-SULFATE
INHIBITOR -> TRANSPORTER
TISSUE EXPRESSION->TRANSPORTER
BASOLATERAL
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: ESTRONE-3-SULFATE
INHIBITOR -> TRANSPORTER
inhibit 30% at 10 μM
IC50
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: Bromsulphthalein (BSP)
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: Bromsulphthalein (BSP)
INHIBITOR -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
INHIBITOR -> TRANSPORTER
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: Estrone 3-sulfate
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: ESTRONE-3-SULFATE
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: Estrone 3-sulfate
INHIBITOR -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
INHIBITOR -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
INHIBITOR -> TRANSPORTER
INHIBITOR -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
SUBSTRATE -> TRANSPORTER
NON-SUBSTRATE -> TRANSPORTER
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: Bromsulphthalein (BSP)
INHIBITOR -> TRANSPORTER
SUBSTRATE USED: Bromsulphthalein
INHIBITOR -> TRANSPORTER
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL