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Showing 41 - 50 of 2,238 results

Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Alletorphine (R & S 218-M) is a potent analgesic said to have a reduced respiratory depressant action. It was isolated by Bentley and Hardy (1967) while they were examining a series of derivatives of tetrahydrothebaine of which the pote...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Ethoxazene (2,4-diamino-4-ethoxyazobenzene) is an analgesic compound. It may be used as an indicator of acidity in an examination of gastric function.
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Imisopasem Manganese is a manganese-based non-peptidyl mimetic of the human mitochondrial manganese superoxide dismutase (MnSOD), with potential antioxidant and radioprotective activities. Metaphore Pharmaceuticals Inc. is developing Imisopasem Mang...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Girisopam (GYKI 51189), a 2,3-benzodiazepine, is a compound with anxiolytic and antipsychotic action. It has shown these effects in several animal models. Girisopam differs from the traditional 1,4-benzodiazepines because of its selective anxiolytic ...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Melizame is a sugar substitute for sweetening caloric or noncaloric materials.
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Evobrutinib is a highly selective, irreversible inhibitor of Bruton's tyrosine kinase (BTK). It potently inhibits BCR- and Fc receptor-mediated signaling and, thus, subsequent activation and function of B cells and innate immune cells such as monocyt...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Emitefur or BOF-A2 is a fluorinated pyrimidine antimetabolite exerting antineoplastic properties. It is a compound composed of 5-fluorouracil (5-FU) and 3-cyano-2,6-dihydroxypyridine (CNDP), an inhibitor of 5-FU degradation by dihydrouracil dehydroge...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)



(-)-3-(3-hydroxyphenyl)-N-n-propylpiperidine ((-)-3-PPP, also known as preclamol) has a dual action towards to dopamine D2 autoreceptor: it activates it and also acts concomitantly as an antagonist at postsynaptic DA receptors. It was shown, that (-)...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

As a narcotic antagonist similar in action to naloxone, DIPRENORPHINE is used to remobilize animals after analgesia by super-potent opioid analgesics such as etorphine and carfentanil. It is not used in humans. Diprenorphine binds approximately equal...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Terbogrel, an agent having two pharmacodynamic actions, namely inhibition of thromboxane A2 synthase and antagonism of the thromboxane A2 receptor. The antithrombotic effect of terbogrel was dose-dependent and was associated with enhanced prostacycli...