Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Sat Dec 16 12:51:23 GMT 2023
by
admin
on
Sat Dec 16 12:51:23 GMT 2023
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
J2234208AE
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
EZH2
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
PRIMARY | |||
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459578-94-0
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
PRIMARY | |||
|
Q15910
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
PRIMARY | |||
|
J2234208AE
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
PRIMARY | |||
|
Q15910
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
PRIMARY | |||
|
487555-47-5
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
ALTERNATIVE | |||
|
EC 2.1.1.43
Created by
admin on Sat Dec 16 12:51:24 GMT 2023 , Edited by admin on Sat Dec 16 12:51:24 GMT 2023
|
PRIMARY |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| O | 1_75 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
biochemical assay
IC50
|
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|
INHIBITOR -> TARGET | |||
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
The maximal dose and schedule attained with GSK2816126 has shown insufficient evidence of clinical activity, and does not justify further clinical investigation.
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) | CHEMICAL |
|