U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:51:23 UTC 2023
Edited
by admin
on Sat Dec 16 12:51:23 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
J2234208AE
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HISTONE-LYSINE N-METHYLTRANSFERASE EZH2
Common Name English
LYSINE N-METHYLTRANSFERASE 6
Common Name English
ENHANCER OF ZESTE 2 (HUMAN CELL LINE BJA-B GENE EZH2)
Common Name English
ENHANCER OF ZESTE HOMOLOG 2
Common Name English
ENX-1
Common Name English
KMT6
Common Name English
Code System Code Type Description
WIKIPEDIA
EZH2
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
PRIMARY
CAS
459578-94-0
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
PRIMARY
UNIPROT
Q15910
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
PRIMARY
FDA UNII
J2234208AE
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
PRIMARY
PHAROS
Q15910
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
PRIMARY
CAS
487555-47-5
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
ALTERNATIVE
EC (ENZYME CLASS)
EC 2.1.1.43
Created by admin on Sat Dec 16 12:51:24 UTC 2023 , Edited by admin on Sat Dec 16 12:51:24 UTC 2023
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
O 1_75
Related Record Type Details
INHIBITOR -> TARGET
biochemical assay
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
The maximal dose and schedule attained with GSK2816126 has shown insufficient evidence of clinical activity, and does not justify further clinical investigation.
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) CHEMICAL