U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Nucleic Acid
Created
by admin
on Wed Apr 02 18:42:38 GMT 2025
Edited
by admin
on Wed Apr 02 18:42:38 GMT 2025
Record UNII
2LVD3H594X
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Cytidine-basivarsen-lysine
Preferred Name English
Code System Code Type Description
FDA UNII
2LVD3H594X
Created by admin on Wed Apr 02 18:42:38 GMT 2025 , Edited by admin on Wed Apr 02 18:42:38 GMT 2025
PRIMARY
Sugar Site Range Site Count
1_1-1_2;1_15-1_16 4 / 16
Deoxyribose (DNA) 1_5-1_12 8 / 16
2'-O-Methoxyethyl ribose 1_3-1_4;1_13-1_14 4 / 16
Linkage Site Range Site Count
Phosporothioate 1_2-1_16 15 / 15

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] 5'-TERMINUS Cytidine-basivarsen-lysine linker 9FC56L2EZB
NUCLEOSIDE BASE SUBSTITUTION [1_15] 5-METHYLCYTOSINE 6R795CQT4H
NUCLEOSIDE BASE SUBSTITUTION [1_14] THYMINE QR26YLT7LT