| Stereochemistry | ACHIRAL |
| Molecular Formula | C25H27N2O5S.Na |
| Molecular Weight | 490.547 |
| Optical Activity | NONE |
| Defined Stereocenters | 0 / 0 |
| E/Z Centers | 0 |
| Charge | 0 |
SHOW SMILES / InChI
SMILES
[Na+].CC(C)(C)C1=CC=C(CN(CC2=CC(OCC([O-])=O)=CC=C2)S(=O)(=O)C3=CN=CC=C3)C=C1
InChI
InChIKey=SVNBMCJEDANCKY-UHFFFAOYSA-M
InChI=1S/C25H28N2O5S.Na/c1-25(2,3)21-11-9-19(10-12-21)16-27(33(30,31)23-8-5-13-26-15-23)17-20-6-4-7-22(14-20)32-18-24(28)29;/h4-15H,16-18H2,1-3H3,(H,28,29);/q;+1/p-1
Evatanepag (CP-533,536) is a prostaglandin E2 EP2 receptor agonist. It stimulates new bone formation on trabecular, endocortical, and periosteal surfaces and enhances fracture healing. Evatanepag was under development with Pfizer as a bone formation stimulant for therapeutic use in the healing of fractures.
Originator
Approval Year
Targets
| Primary Target | Pharmacology | Condition | Potency |
|---|---|---|---|
| 5.0 nM [EC50] |
PubMed
Patents
ACTIVE MOIETY
SUBSTANCE RECORD
