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Showing 11 - 20 of 116 results

Status:
US Approved Rx (2022)
First approved in 1985

Class (Stereo):
CHEMICAL (RACEMIC)



Mexiletine is a non-selective voltage-gated sodium channel blocker which belongs to the Class IB anti-arrhythmic group of medicines. It is used to treat heart arrhythmias. Mexiletine is also used to treat refractory pain and muscle stiffness resultin...
Status:
US Approved Rx (2000)
First approved in 1984

Class (Stereo):
CHEMICAL (ACHIRAL)



Inamrinone (Amrinone) is a positive inotropic cardiotonic with vasodilator properties, phosphodiesterase inhibitory activity, and the ability to stimulate calcium ion influx into the cardiac cell. Inamrinone is a phosphodiesterase inhibitor (PDE3), r...
Status:
US Approved Rx (1998)
First approved in 1981

Class (Stereo):
CHEMICAL (ABSOLUTE)



Ecraprost [AS 013, Circulase] is a prodrug of prostaglandin E(1) within lipid microspheres that is being developed in Japan by Mitsubishi Pharma Corporation and Asahi Glass. It was originally in development with Welfide Corporation. On 1 October 2001...
Status:
US Approved Rx (1993)
First approved in 1978

Class (Stereo):
CHEMICAL (RACEMIC)


Conditions:

Dobutamine is a sympathomimetic drug used in the treatment of heart failure and cardiogenic shock. Dobutamine hydrochloride is a direct-acting inotropic agent whose primary activity results from stimulation of the ß-receptors of the heart while produ...
Status:
US Approved Rx (1985)
First approved in 1977

Class (Stereo):
CHEMICAL (RACEMIC)



Disopyramide is an antiarrhythmic drug indicated for the treatment of documented ventricular arrhythmias, such as sustained ventricular tachycardia that are life-threatening. In man, Disopyramide at therapeutic plasma levels shortens the sinus node r...
Status:
US Approved Rx (2020)
First approved in 1974

Class (Stereo):
CHEMICAL (RACEMIC)



Ibuprofen is a nonsteroidal anti-inflammatory agent (NSAIA) or nonsteroidal anti-inflammatory drug (NSAID), with analgesic and antipyretic properties. Ibuprofen has pharmacologic actions similar to those of other prototypical NSAIAs, which are though...
Status:
US Approved Rx (2018)
First approved in 1974

Class (Stereo):
CHEMICAL (ACHIRAL)



Dopamine, a sympathomimetic amine vasopressor, is the naturally occurring immediate precursor of norepinephrine. G protein-coupled dopamine receptors (D1, D2, D3, D4, and D5) mediate all of the physiological functions of the catecholaminergic neurotr...
Status:
US Approved Rx (2010)
First approved in 1965

Class (Stereo):
CHEMICAL (ACHIRAL)



Indometacin (INN and BAN) or indomethacin (AAN, USAN, and former BAN) is a nonsteroidal anti-inflammatory drug (NSAID) commonly used as a prescription medication to reduce fever, pain, stiffness, and swelling from inflammation. Indomethacin has analg...
Status:
US Approved Rx (2002)
First approved in 1954

Class (Stereo):
CHEMICAL (ABSOLUTE)



Digoxin, a cardiac glycoside similar to digitoxin, is used to treat congestive heart failure and supraventricular arrhythmias due to reentry mechanisms, and to control ventricular rate in the treatment of chronic atrial fibrillation. Digoxin inhibits...
Status:
US Approved Rx (2021)
First approved in 1954

Class (Stereo):
CHEMICAL (ABSOLUTE)



Metaraminol is a potent sympathomimetic amine that increases both systolic and diastolic blood pressure, is an adrenergic receptor alpha-1 agonist.. Metaraminol is indicated for prevention and treatment of the acute hypotensive state occurring with s...

Showing 11 - 20 of 116 results