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Showing 111 - 120 of 612 results

Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Mecloqualone is a quinazoline-class GABAergic and an analog of methaqualone. It acts as an agonist of the beta subtype of GABAa receptor and induces sedative, hypnotic and anxiolytic effects. Mecloqualone was marketed (mostly in france) under the nam...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Myrophine is an opiate analog and long-acting prodrug for morphine with a slow onset of effects. It is weaker than morphine as an analgesic but longer-lasting in effects and was thought to have a more local anesthetic effect than morphine, though wit...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Eticyclidine (N-ethyl-1-phenylcyclohexylamine) is a phencyclidine derivative exerting nearly the same pharmacological profile as the parent compound. In rodents, it induces stereotypy, ataxia, interoceptive effect and hypothermia.
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)


Conditions:

Desomorphine is the common name for 4,5--epoxy-17- methylmorphinan-3-ol or dihydrodesoxymorphine-D. It is an opioid analogue and morphine derivative in which the 6-hydroxyl group and the double bond at carbons 7 and 8 of morphine are reduced. Desomor...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Conditions:

Etonitazene is a potent and selective mu-opioid agonist. It was developed in CIBA. Administration of etonitazene may induce respiratory depression, and therefor etonitazene is not used in humans. Etonitazene is explicitly listed as an illegal drug un...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Carfentanil is a synthetic fentanyl analog. It is a mu-opioid receptor agonist with an estimated analgesic potency approximately 10,000 times that of morphine and 20-30 times that of fentanyl, based on animal studies. Receptor binding studies have s...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Benzethidine an opioid analgesic that was forbidden for use.
Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)

Betaprodine is an opioid analgesic under international control according to the UN Single Convention 1961. It has been used in obstetrics, as pre-operative medication, for minor surgical procedures.
Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)

Diampromide is a synthetic narcotic analgesic. It was designed as a methadone analog and hence with a chiral center similar to that of the parent. Diampromide approximates to the potency of pethidine and morphine in mice and rats, respectively. It ha...
Status:
Investigational

Class (Stereo):
CHEMICAL (MIXED)

Proheptazine is a substituted azacycloalkane patented by American Home Products Corp. as an opioid analgesic. Proheptazine produces similar effects to other opioids, including analgesia, sedation, euphoria, dizziness and nausea.

Showing 111 - 120 of 612 results