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Status:
US Approved Rx (2022)
First approved in 2003

Class (Stereo):
CHEMICAL (ACHIRAL)



Gefitinib is an anilinoquinazoline with antineoplastic activity. Gefitinib inhibits the epidermal growth factor receptor (EGFR) tyrosine kinase by binding to the adenosine triphosphate (ATP)-binding site of the enzyme. Thus the function of the EGFR t...