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Showing 11 - 20 of 35 results

Androstanol is a steroid acting as the inverse agonist of constitutive androstane receptor. In addition, androstanol activates pregnane X receptor. In animal models, it protects from drug-induced liver injury. Androstanol appears to be a pheromone.
Status:
Other

Class (Stereo):
CHEMICAL (ABSOLUTE)


Conditions:

(3S,5R)-atorvastatin is a stereoisomer of atorvastatin. Atorvastatin is a synthetic hydroxymethylglutaryl coenzyme A (HMG-CoA) reductase inhibitor. 3R,5R enantiopure form of atorvastatin (Lipitor, Pfizer; since Nov 2011 generic) is used clinically. I...
Ginkgolide A (GA, BN52020), is a terpene lactone constituent of Ginkgo biloba, the ginkgo tree, is the oldest living tree, with a long history of use in traditional Chinese medicine. Ginkgolide A is an effective antagonist of platelet activating fact...
Guggulsterone is a naturally occuring bioactive plant sterol isolated from the gum resin of guggul (Commiphora wightii), which potently reverses multi-drug resistance in a number of human cancer cell lines, extending the efficacy of chemotherapy. Gug...
Flavonol (3-Hydroxyflavone) is a practically insole synthetic compound, which is not found naturally in plants. 3-hydroxyflavone can be found in a number of food items such as brassicas, pomegranate, red raspberry, and fenugreek, which makes 3-hydrox...
Status:
Possibly Marketed Outside US
First approved in 2013

Class (Stereo):
CHEMICAL (ABSOLUTE)



Zeranol is a non-steroidal anabolic growth promoter with potent estrogenic activity that is widely used as a growth promoter in the US beef industry. It is a mycotoxin, derived from fungi in the Fusarium family, it is an estrogen agonist. Zeranol is...
Status:
Possibly Marketed Outside US
First approved in 2013

Class (Stereo):
CHEMICAL (ABSOLUTE)



Stevioside, an abundant component of Stevia rebaudiana leaf, has become well-known for its intense sweetness (250-300 times sweeter than sucrose) and is used as a non-caloric sweetener in several countries. Steviol and isosteviol (metabolic component...
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (RACEMIC)



Flutrimazole (trade names Flusporan, Funcenal, Micetal, Topiderm) is an imidazole derivative, a wide-spectrum antifungal drug used for the topical treatment of superficial mycoses of the skin. Flutrimazole interferes with the synthesis of ergosterol ...
Status:
US Approved Rx (2014)
First approved in 2004

Class (Stereo):
CHEMICAL (ACHIRAL)



Erlotinib hydrochloride (trade name Tarceva, Genentech/OSIP, originally coded as OSI-774) is a drug used to treat non-small cell lung cancer, pancreatic cancer and several other types of cancer. Similar to gefitinib, erlotinib specifically targets th...

Showing 11 - 20 of 35 results