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Showing 1 - 10 of 10 results

Status:
US Approved Rx (2000)
First approved in 2000

Class (Stereo):
CHEMICAL (ABSOLUTE)



Cetrorelix is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH) from the gonadotrophic cells of the ant...
Status:
US Approved Rx (1993)
First approved in 1985

Class (Stereo):
CHEMICAL (ABSOLUTE)



Leuprolide acetate is a synthetic nonapeptide analog of naturally occurring gonadotropin-releasing hormone (GnRH or LH-RH). The analog possesses greater potency than the natural hormone. It acts primarily on the anterior pituitary, inducing a transie...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)



Zibotentan (ZD4054) is a potent and specific orally available endothelin A (ETA) receptor antagonist, with no measurable affinity for endothelin B receptor. Activation of the ETA receptor by ET-1 has emerged as an important factor promoting tumor cel...
Status:
US Previously Marketed
First approved in 2003

Class (Stereo):
CHEMICAL (ABSOLUTE)



Abarelix is a synthetic decapeptide antagonist to gonadotropin releasing hormone (GnRH). It is marketed by Praecis Pharmaceuticals as Plenaxis. Used in the palliative treatment of advanced prostate cancer. Abarelix is a luteinizing hormone agonist t...
Status:
US Approved Rx (2000)
First approved in 2000

Class (Stereo):
CHEMICAL (ABSOLUTE)



Cetrorelix is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH) from the gonadotrophic cells of the ant...
Status:
US Approved Rx (2000)
First approved in 2000

Class (Stereo):
CHEMICAL (ABSOLUTE)



Cetrorelix is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH) from the gonadotrophic cells of the ant...
Status:
US Approved Rx (2000)
First approved in 2000

Class (Stereo):
CHEMICAL (ABSOLUTE)



Cetrorelix is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH) from the gonadotrophic cells of the ant...
Status:
US Approved Rx (2000)
First approved in 2000

Class (Stereo):
CHEMICAL (ABSOLUTE)



Cetrorelix is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH) from the gonadotrophic cells of the ant...
Status:
US Approved Rx (1993)
First approved in 1985

Class (Stereo):
CHEMICAL (ABSOLUTE)



Leuprolide acetate is a synthetic nonapeptide analog of naturally occurring gonadotropin-releasing hormone (GnRH or LH-RH). The analog possesses greater potency than the natural hormone. It acts primarily on the anterior pituitary, inducing a transie...
Status:
US Approved Rx (1993)
First approved in 1985

Class (Stereo):
CHEMICAL (ABSOLUTE)



Leuprolide acetate is a synthetic nonapeptide analog of naturally occurring gonadotropin-releasing hormone (GnRH or LH-RH). The analog possesses greater potency than the natural hormone. It acts primarily on the anterior pituitary, inducing a transie...