U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

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Status:
Investigational
Source:
INN:cartazolate [INN]
Source URL:

Class (Stereo):
CHEMICAL (ACHIRAL)

Cartazolate (also known as SQ-65,396) is GABAA receptor positive allosteric modulator with potent anxiolytic activity proven in clinical trials. Cartazolate is also known to act as an adenosine antagonist at the A1 and A2 subtypes and as a phosphodiesterase inhibitor.