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Showing 11 - 20 of 20 results

Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (EPIMERIC)

Acrocinonide (or triamcinolone acroleinide) a glucocorticoid anti-inflammatory compound, which has never been marketed.
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)


Piquizil, a 4-aminoquinazoline causing relaxation of respiratory smooth muscle in animals, appeared to be a bronchodilator in man. It has been shown to be equal in activity to a combination of theophylline, ephedrine and phenobarbital. Piquizil and T...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Tetrazolast (also known as MDL 26,024GO) is a tetrazoloquinoline derivative patented by Merrell Dow Pharmaceuticals, Inc. as an antiallergic and antiasthmatic agent. Tetrazolast was shown to be an orally absorbed mediator release inhibitor in the rat...
Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)

Metalol is an antagonist at beta-adrenergic receptors.
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Butoprozine increased the action potential duration like amiodarone, depressed the plateau phase like verapamil and decreased the amplitude and the maximum rate of depolarization. Butoprozine injected intravenously depressed sino-atrial node functio...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Tetrazolast (also known as MDL 26,024GO) is a tetrazoloquinoline derivative patented by Merrell Dow Pharmaceuticals, Inc. as an antiallergic and antiasthmatic agent. Tetrazolast was shown to be an orally absorbed mediator release inhibitor in the rat...
Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)


Tazolol is a selective myocardial beta-blocking agent. Experiments on dogs have shown that this compound could be useful in patients with heart failure due to coronary artery disease. However, information about the current use of tazolol is not avail...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)


Levophacetoperane is a piperidine derivative. Levofacetoperane is a sympathomimetic central nervous system stimulant and is commonly used to treat depression. Levophacetoperane is also a known analeptic and is strongly linked to apnea reversal in dog...
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (RACEMIC)


Pipoxolan is an antispasmodic drug. In vivo, the drug inhibited the contractions of intestines caused by neostigmine, barium chloride or injection of acetylcholine. The drug possesses ganglioplegic action and inhibited the decrease in blood pressure ...
Status:
Possibly Marketed Outside US

Class (Stereo):
CHEMICAL (ACHIRAL)

Clamoxyquin is an antiamebic and antidiarrheal agent. Clamoxyquin is usually used as the pamoate or hydrochloride salt. It is a veterinary antiparasitic drug used to treat salmonids for the myxozoan parasite Myxobolus cerebralis. Dietary inclusion o...

Showing 11 - 20 of 20 results