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XORPHANOL

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  L415991P58

Status:
Investigational
Source:
INN:xorphanol
Source URL:
https://tripod.nih.gov/npc/#Download
Class (Stereo):
CHEMICAL (ABSOLUTE)
Xorphanol (also known as TR5379M) is a full κ-opioid receptor agonist and is a partial agonist at μ opioid receptor. Clinically, xorphanol was studied as an orally active analgesic that provided effective pain relief but showed low physical dependence liability. Further development of this drug was discontinued.

XORPHANOL MESYLATE

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  A88BIS7IBB

Status:
Investigational
Source:
INN:xorphanol
Source URL:
https://tripod.nih.gov/npc/#Download
Class (Stereo):
CHEMICAL (ABSOLUTE)
Xorphanol (also known as TR5379M) is a full κ-opioid receptor agonist and is a partial agonist at μ opioid receptor. Clinically, xorphanol was studied as an orally active analgesic that provided effective pain relief but showed low physical dependence liability. Further development of this drug was discontinued.
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NCATS
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