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Showing 1 - 3 of 3 results

Status:
Investigational

Class (Stereo):
CHEMICAL (RACEMIC)

Cicloprofen is fluorene derivative patented by American pharmaceutical company E. R. Squibb as anti-inflammatory agents. Cicloprofen is potent cyclooxygenase inhibitor. Cicloprofen undergoes hydroxylation of the fluorene rings and conjugation with gl...
Status:
Investigational

Class (Stereo):
CHEMICAL (ABSOLUTE)

Ceronapril is a phosphonate angiotensin-converting enzyme inhibitor that was being developed by Bristol-Myers Squibb for the treatment of hypertension. In spontaneously hypertensive rats, Ceronapril narrowed the autoregulatory range and shifted it to...
Status:
Investigational

Class (Stereo):
CHEMICAL (ACHIRAL)

Cartazolate (also known as SQ-65,396) is GABAA receptor positive allosteric modulator with potent anxiolytic activity proven in clinical trials. Cartazolate is also known to act as an adenosine antagonist at the A1 and A2 subtypes and as a phosphod...