U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 05:17:49 GMT 2025
Edited
by admin
on Wed Apr 02 05:17:49 GMT 2025
Protein Type BISPECIFIC ANTIBODY
Protein Sub Type
Sequence Type COMPLETE
Record UNII
ZR1EEO1ZLS
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
VEPSITAMAB
INN  
Official Name English
IMMUNOGLOBULIN, BISPECIFIC, ANTI-(HUMAN MUCIN 17) (HUMAN MONOCLONAL MUC17_CD3_ALT2 SINGLE-CHAIN VARIABLE FRAGMENT VH1-(GGGGS)3-VL1) FUSION PROTEIN WITH PEPTIDE LINKER (GGGGS) FUSION PROTEIN WITH IMMUNOGLOBULIN ANTI-(HUMAN CD3 ANTIGEN .EPSILON.-CHAIN) (HU
Preferred Name English
vepsitamab [INN]
Common Name English
Vepsitamab [WHO-DD]
Common Name English
Classification Tree Code System Code
FDA ORPHAN DRUG 741120
Created by admin on Wed Apr 02 05:17:49 GMT 2025 , Edited by admin on Wed Apr 02 05:17:49 GMT 2025
Code System Code Type Description
INN
11822
Created by admin on Wed Apr 02 05:17:49 GMT 2025 , Edited by admin on Wed Apr 02 05:17:49 GMT 2025
PRIMARY
SMS_ID
300000009420
Created by admin on Wed Apr 02 05:17:49 GMT 2025 , Edited by admin on Wed Apr 02 05:17:49 GMT 2025
PRIMARY
FDA UNII
ZR1EEO1ZLS
Created by admin on Wed Apr 02 05:17:49 GMT 2025 , Edited by admin on Wed Apr 02 05:17:49 GMT 2025
PRIMARY
CAS
2413453-53-7
Created by admin on Wed Apr 02 05:17:49 GMT 2025 , Edited by admin on Wed Apr 02 05:17:49 GMT 2025
PRIMARY
NCI_THESAURUS
C165588
Created by admin on Wed Apr 02 05:17:49 GMT 2025 , Edited by admin on Wed Apr 02 05:17:49 GMT 2025
PRIMARY
From To
1_22 1_95
1_44 1_234
1_157 1_222
1_269 1_345
1_409 1_477
1_506 1_763
1_509 1_766
1_541 1_601
1_572 1_582
1_647 1_705
1_798 1_858
1_829 1_839
1_904 1_962
Related Record Type Details
ACTIVE MOIETY

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID REMOVAL [1_984] C-TERMINUS LYSINE K3Z4F929H6
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL