U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 14:32:18 GMT 2025
Edited
by admin
on Wed Apr 02 14:32:18 GMT 2025
Protein Type RECEPTOR
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
UUW939U56A
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Nischarin
Common Name English
I1-Imidazoline Receptor
Preferred Name English
Imidazoline-1 receptor
Common Name English
Imidazoline receptor 1
Common Name English
Code System Code Type Description
FDA UNII
UUW939U56A
Created by admin on Wed Apr 02 14:32:18 GMT 2025 , Edited by admin on Wed Apr 02 14:32:18 GMT 2025
PRIMARY
Related Record Type Details
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
Ki
AGONIST -> TARGET
Ki
AGONIST -> TARGET
AGONIST -> TARGET
Ki
AGONIST -> TARGET
Ki

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_540] [1_542] [1_545] [1_1021] [1_1283] SITE_SPECIFIC S DEXFOSFOSERINE VI4F0K069V
AMINO_ACID_SUBSTITUTION [1_1] SITE_SPECIFIC A N-ACETYLALANINE 26C4VY6Z0M
AMINO_ACID_SUBSTITUTION [1_1281] SITE_SPECIFIC T THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL