U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 01:20:22 GMT 2025
Edited
by admin
on Wed Apr 02 01:20:22 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
SV6QS63US6
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
C-C CHEMOKINE RECEPTOR TYPE 1
Common Name English
C-C CKR-1
Preferred Name English
CD191
Common Name English
RANTES-R
Common Name English
CMKBR1
Common Name English
CMKR1
Common Name English
MACROPHAGE INFLAMMATORY PROTEIN 1-ALPHA RECEPTOR
Common Name English
CCR1
Common Name English
MIP-1ALPHA-R
Common Name English
LD78 RECEPTOR
Common Name English
HM145
Common Name English
CCR-1
Common Name English
SCYAR1
Common Name English
Code System Code Type Description
FDA UNII
SV6QS63US6
Created by admin on Wed Apr 02 01:20:22 GMT 2025 , Edited by admin on Wed Apr 02 01:20:22 GMT 2025
PRIMARY
UNIPROT
P32246
Created by admin on Wed Apr 02 01:20:22 GMT 2025 , Edited by admin on Wed Apr 02 01:20:22 GMT 2025
PRIMARY
From To
1_106 1_183
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_5
Related Record Type Details
INHIBITOR -> TARGET
Efficacious in multiple myeloma in preclinical but ineffective in phase II clinical trials for multiple sclerosis.
Ki
INHIBITOR -> TARGET
Compound Inhibited recruitment of immune cells induced by CCL3, but a phase II trial investigating rheumatoid arthritis was terminated due to no discernible activity in patients with rheumatoid arthritis at a concentration of 10 mg once daily.
INHIBITOR -> TARGET
Binding Assay
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Binding assay
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_340] [1_341] [1_345] [1_352] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL