U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
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Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:17:53 GMT 2025
Edited
by admin
on Tue Apr 01 18:17:53 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
RWA84PTK5G
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ANTIGEN NY-CO-9
Preferred Name English
HISTONE DEACETYLASE 5
Common Name English
HD5
Common Name English
HDAC5
Common Name English
KIAA0600
Common Name English
Code System Code Type Description
FDA UNII
RWA84PTK5G
Created by admin on Tue Apr 01 18:17:53 GMT 2025 , Edited by admin on Tue Apr 01 18:17:53 GMT 2025
PRIMARY
UNIPROT
Q9UQL6
Created by admin on Tue Apr 01 18:17:53 GMT 2025 , Edited by admin on Tue Apr 01 18:17:53 GMT 2025
PRIMARY
WIKIPEDIA
Histone deacetylase 5
Created by admin on Tue Apr 01 18:17:53 GMT 2025 , Edited by admin on Tue Apr 01 18:17:53 GMT 2025
PRIMARY
PHAROS
Q9UQL6
Created by admin on Tue Apr 01 18:17:53 GMT 2025 , Edited by admin on Tue Apr 01 18:17:53 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
Pan HDAC inhibitor
NON-INHIBITOR->TARGET
WEAK INHIBITOR->TARGET
BINDING
IC50
WEAK INHIBITOR->TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_259] [1_661] [1_1108] DEXFOSFOSERINE VI4F0K069V
AMINO_ACID_SUBSTITUTION [1_533] N6-ACETYLLYSINE 470AD5VY1X
AMINO_ACID_SUBSTITUTION [1_292] THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL