U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 06:12:31 GMT 2025
Edited
by admin
on Wed Apr 02 06:12:31 GMT 2025
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG1
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
RAQ1MR035D
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PELGIFATAMAB
INN  
Official Name English
IMMUNOGLOBULIN G1, ANTI-(HUMAN PROSTATE-SPECIFIC MEMBRANE ANTIGEN) (HUMAN MONOCLONAL TPP-7195 .GAMMA.1-CHAIN), DISULFIDE WITH HUMAN MONOCLONAL TPP-7195 .KAPPA.-CHAIN, DIMER
Preferred Name English
pelgifatamab [INN]
Common Name English
Code System Code Type Description
NCI_THESAURUS
C203129
Created by admin on Wed Apr 02 06:12:31 GMT 2025 , Edited by admin on Wed Apr 02 06:12:31 GMT 2025
PRIMARY
CAS
2414550-93-7
Created by admin on Wed Apr 02 06:12:31 GMT 2025 , Edited by admin on Wed Apr 02 06:12:31 GMT 2025
PRIMARY
SMS_ID
300000046959
Created by admin on Wed Apr 02 06:12:31 GMT 2025 , Edited by admin on Wed Apr 02 06:12:31 GMT 2025
PRIMARY
INN
11920
Created by admin on Wed Apr 02 06:12:31 GMT 2025 , Edited by admin on Wed Apr 02 06:12:31 GMT 2025
PRIMARY
FDA UNII
RAQ1MR035D
Created by admin on Wed Apr 02 06:12:31 GMT 2025 , Edited by admin on Wed Apr 02 06:12:31 GMT 2025
PRIMARY
From To
1_22 1_96
2_22 2_96
2_150 2_206
2_226 4_214
2_267 2_327
1_150 1_206
2_373 2_431
3_23 3_88
3_134 3_194
4_23 4_88
4_134 4_194
1_226 3_214
1_232 2_232
1_235 2_235
1_267 1_327
1_373 1_431
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_303
N 2_303

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] [2_1] N-TERMINUS Q PIDOLIC ACID SZB83O1W42
AMINO ACID REMOVAL [1_453] [2_453] C-TERMINUS Amount: LYSINE K3Z4F929H6
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL