Details
| Stereochemistry | RACEMIC |
| Molecular Formula | C21H30N4O4 |
| Molecular Weight | 402.4873 |
| Optical Activity | ( + / - ) |
| Defined Stereocenters | 0 / 1 |
| E/Z Centers | 0 |
| Charge | 0 |
SHOW SMILES / InChI
SMILES
CCOC1=C(C=C(C(N)=C1)[N+]([O-])=O)C(=O)NC2CCN(CC3CCC=CC3)CC2
InChI
InChIKey=ZDLBNXXKDMLZMF-UHFFFAOYSA-N
InChI=1S/C21H30N4O4/c1-2-29-20-13-18(22)19(25(27)28)12-17(20)21(26)23-16-8-10-24(11-9-16)14-15-6-4-3-5-7-15/h3-4,12-13,15-16H,2,5-11,14,22H2,1H3,(H,23,26)
| Molecular Formula | C21H30N4O4 |
| Molecular Weight | 402.4873 |
| Charge | 0 |
| Count |
|
| Stereochemistry | RACEMIC |
| Additional Stereochemistry | No |
| Defined Stereocenters | 0 / 1 |
| E/Z Centers | 0 |
| Optical Activity | ( + / - ) |
Cinitapride is an agonist of 5-HT4 and 5-HT1 receptors and antagonist of 5-HT2 receptors. Cinitapride is marketed worldwide for the treatment of gastrointestinal disorders related to motility such as indigestion or functional or non-ulcer dyspepsia, gastroesophageal reflux diseases, delay in gastric emptying and vomiting.
Approval Year
PubMed
| Title | Date | PubMed |
|---|---|---|
| [Efficacy and tolerance of cinitapride on the disturbances of gastrointestinal transit]. | 1991 Jul-Sep |
|
| Cinitapride protects against ethanol-induced gastric mucosal injury in rats: role of 5-hydroxytryptamine, prostaglandins and sulfhydryl compounds. | 1997 Apr |
|
| Effects of cinitapride on gastric ulceration and secretion in rats. | 1998 Mar |
| Substance Class |
Chemical
Created
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R8I97I2L24
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| Record Status |
Validated (UNII)
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A03FA08
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C66885
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C47794
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100000081046
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C77257
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m3565
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CINITAPRIDE
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C045316
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21125
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DTXSID60867232
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DB08810
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| Related Record | Type | Details | ||
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ENANTIOMER -> RACEMATE | |||
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ENANTIOMER -> RACEMATE | |||
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TARGET -> INHIBITOR |
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ACTIVE MOIETY |
