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Details

Stereochemistry ACHIRAL
Molecular Formula C15H7F7NO3.Na
Molecular Weight 405.1996
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of NELONEMDAZ SODIUM

SMILES

[Na+].OC1=C(C=C(NCC2=C(F)C(F)=C(C(F)=C2F)C(F)(F)F)C=C1)C([O-])=O

InChI

InChIKey=JRUKCFQBEJZBGU-UHFFFAOYSA-M
InChI=1S/C15H8F7NO3.Na/c16-10-7(11(17)13(19)9(12(10)18)15(20,21)22)4-23-5-1-2-8(24)6(3-5)14(25)26;/h1-3,23-24H,4H2,(H,25,26);/q;+1/p-1

HIDE SMILES / InChI

Molecular Formula C15H7F7NO3
Molecular Weight 382.2098
Charge -1
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Molecular Formula Na
Molecular Weight 22.98976928
Charge 1
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

PubMed

PubMed

TitleDatePubMed
Neu2000, an NR2B-selective, moderate NMDA receptor antagonist and potent spin trapping molecule for stroke.
2010-11
The functional and neuroprotective actions of Neu2000, a dual-acting pharmacological agent, in the treatment of acute spinal cord injury.
2010-01
The novel NMDA receptor antagonist, 2-hydroxy-5-(2,3,5,6-tetrafluoro-4-trifluoromethyl-benzylamino)-benzoic acid, is a gating modifier in cultured mouse cortical neurons.
2009-06
Marked prevention of ischemic brain injury by Neu2000, an NMDA antagonist and antioxidant derived from aspirin and sulfasalazine.
2007-06
Concurrent administration of Neu2000 and lithium produces marked improvement of motor neuron survival, motor function, and mortality in a mouse model of amyotrophic lateral sclerosis.
2007-04
Patents
Substance Class Chemical
Created
by admin
on Tue Apr 01 16:30:41 GMT 2025
Edited
by admin
on Tue Apr 01 16:30:41 GMT 2025
Record UNII
MMY7F8FR6C
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
NEU-2000 SODIUM SALT
Preferred Name English
NELONEMDAZ SODIUM
Common Name English
BENZOIC ACID, 2-HYDROXY-5-(((2,3,5,6-TETRAFLUORO-4-(TRIFLUOROMETHYL)PHENYL)METHYL)AMINO)-, SODIUM SALT (1:1)
Systematic Name English
2-HYDROXY-5-((2,3,5,6-TETRAFLUORO-4-(TRIFLUOROMETHYL)PHENYL)METHYLAMINO)BENZOIC ACID, SODIUM HYDRIDE
Systematic Name English
Code System Code Type Description
FDA UNII
MMY7F8FR6C
Created by admin on Tue Apr 01 16:30:41 GMT 2025 , Edited by admin on Tue Apr 01 16:30:41 GMT 2025
PRIMARY
PUBCHEM
23666512
Created by admin on Tue Apr 01 16:30:41 GMT 2025 , Edited by admin on Tue Apr 01 16:30:41 GMT 2025
PRIMARY
CAS
916214-58-9
Created by admin on Tue Apr 01 16:30:41 GMT 2025 , Edited by admin on Tue Apr 01 16:30:41 GMT 2025
PRIMARY
Related Record Type Details
PARENT -> SALT/SOLVATE
Related Record Type Details
ACTIVE MOIETY