U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:00:55 UTC 2023
Edited
by admin
on Sat Dec 16 12:00:55 UTC 2023
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
M8873UUY31
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HISTONE DEACETYLASE 11
Common Name English
HDAC11
Common Name English
Code System Code Type Description
UNIPROT
Q96DB2
Created by admin on Sat Dec 16 12:00:55 UTC 2023 , Edited by admin on Sat Dec 16 12:00:55 UTC 2023
PRIMARY
FDA UNII
M8873UUY31
Created by admin on Sat Dec 16 12:00:55 UTC 2023 , Edited by admin on Sat Dec 16 12:00:55 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Enzymatic Inhibition
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
Enzymatic Inhibition
IC50
INHIBITOR -> TARGET
Mocetinostat (MGCD0103) is a potent HDAC inhibitor with a 2- to 10- fold selectivity against HDAC11. Phase 2.
INHIBITOR
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL