PIPERACETAZINE

Details

Stereochemistry	ACHIRAL
Molecular Formula	C24H30N2O2S
Molecular Weight	410.572
Optical Activity	NONE
Defined Stereocenters	0 / 0
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure Search

SMILES

CC(=O)C1=CC=C2SC3=C(C=CC=C3)N(CCCN4CCC(CCO)CC4)C2=C1

InChI

InChIKey=BTFMCMVEUCGQDX-UHFFFAOYSA-N

InChI=1S/C24H30N2O2S/c1-18(28)20-7-8-24-22(17-20)26(21-5-2-3-6-23(21)29-24)13-4-12-25-14-9-19(10-15-25)11-16-27/h2-3,5-8,17,19,27H,4,9-16H2,1H3

HIDE SMILES / InChI

Molecular Formula	C24H30N2O2S
Molecular Weight	410.572
Charge	0
Count

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Description
Sources: http://ajp.psychiatryonline.org/doi/abs/10.1176/ajp.120.9.900

Piperacetazine (Quide) is an antipsychotic prodrug, most notably used for schizophrenia. The study indicates that Quide is a useful addition to the armamentarium of the physician faced with the difficult problem of treating the chronic hospitalized patient with a schizophrenic illness. Side effects of the drug were generally mild, and there was no evidence that it would produce blood dyscrasias or liver impairment.

Originator

Approval Year

Conditions

Condition	Modality	Targets	Highest Phase	Product
Chronic schizophrenia 6 Sources: http://ajp.psychiatryonline.org/doi/abs/10.1176/ajp.120.9.900	Primary		Approved 8429	QUIDE Approved Use Piperacetazine Launch Date 1969

Sourcing

Vendor/Aggregator	ID	URL
001 Chemical	DY552254	https://www.001chemical.com/chem/3819-00-9
AA Blocks	AA00C6GW	https://www.aablocks.com/goods/Goods/detail?id=AA00C6GW
Aaron Chemicals	AR00C78O	http://www.aaronchem.com/3819-00-9
Ambinter	Amb22731584	http://www.ambinter.com/reference/22731584
Angel Pharmatech	AG-19986	http://www.angelpharmatech.com/3819-00-9.html
Aurora Fine Chemicals LLC	A17.945.941	http://online.aurorafinechemicals.com/info?ID=A17.945.941
BLD Pharm	BD148123	http://www.bldpharm.com/products/3819-00-9.html
CSNpharm	CSN11726	https://www.csnpharm.com/products/piperacetazine.html
Chem Scene	CS-4756	http://www.chemscene.com/3819-00-9.html
ChemMol	99085604	http://www.chemmol.com/chemmol/99085604.html
Chemspace	CSSB00000734558	https://chem-space.com/CSSB00000734558
Enamine	Z2065671295	https://www.enaminestore.com/catalog/Z2065671295
Hairui	HR100562	http://www.hairuichem.com/en/product/3819-00-9.html
LGC Standards	LGCFOR3212.00	https://www.lgcstandards.com/US/en/p/LGCFOR3212.00
LGC Standards	MM3212.00	https://www.lgcstandards.com/US/en/p/MM3212.00
MedChem Express	HY-B1152	https://www.medchemexpress.com/Piperacetazine.html
Molcore	MC552254	https://www.molcore.com/product/3819-00-9
MuseChem	I003403	https://www.musechem.com/product/I003403.html
OChem	30688	http://www.ocheminc.com/index.php?act=psearch&pid=819P009
Sigma-Aldrich	PH004722_ALDRICH	https://www.sigmaaldrich.com/catalog/product/aldrich/ph004722
Smolecule	S539730	http://www.smolecule.com/products/s539730
THE BioTek	bt-278569	https://www.thebiotek.com/product/inhibitors/bt-278569
eNovation Chemicals	D671341	https://www.enovationchem.com/ProductDetails.asp?ProductID=D671341
eNovation Chemicals	D963429	https://www.enovationchem.com/ProductDetails.asp?ProductID=D963429

PubMed

Title	Date	PubMed
Atypical tardive dyskinesia.	1975 May	1119614

Patents

Sample Use Guides

In Vivo Use Guide

Unknown

Route of Administration: Oral

In Vitro Use Guide

Unknown

Substance Class	Chemical Created by `admin` on `Fri Dec 15 15:04:11 GMT 2023` Edited by `admin` on `Fri Dec 15 15:04:11 GMT 2023`
Record UNII	KL6248WNW4
Record Status	`Validated (UNII)`
Record Version

Download

Name

Type

Language

PIPERACETAZINE

Official Name

English

PIPERACETAZINE [ORANGE BOOK]

Common Name

English

NSC-760067

Code

English

QUIDE

Brand Name

English

PIPERACETAZINE [GREEN BOOK]

Common Name

English

PC-1421

Code

English

PIPERACETAZINE [VANDF]

Common Name

English

Piperacetazine [WHO-DD]

Common Name

English

10-[3-[4-(2-Hydroxyethyl)piperidino]propyl]phenothiazin-2-yl methyl ketone

Systematic Name

English

PIPERACETAZINE [MI]

Common Name

English

ETHANONE, 1-(10-(3-(4-(2-HYDROXYETHYL)-1-PIPERIDINYL)PROPYL)-10H-PHENOTHIAZIN-2-YL)-

Systematic Name

English

PIPERACETAZINE [MART.]

Common Name

English

PIPERACETAZINE [USAN]

Common Name

English

piperacetazine [INN]

Common Name

English

Classification Tree Code System Code

NCI_THESAURUS

C740