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Details

Stereochemistry ACHIRAL
Molecular Formula C24H30N2O2S
Molecular Weight 410.572
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of PIPERACETAZINE

SMILES

CC(=O)C1=CC=C2SC3=C(C=CC=C3)N(CCCN4CCC(CCO)CC4)C2=C1

InChI

InChIKey=BTFMCMVEUCGQDX-UHFFFAOYSA-N
InChI=1S/C24H30N2O2S/c1-18(28)20-7-8-24-22(17-20)26(21-5-2-3-6-23(21)29-24)13-4-12-25-14-9-19(10-15-25)11-16-27/h2-3,5-8,17,19,27H,4,9-16H2,1H3

HIDE SMILES / InChI

Molecular Formula C24H30N2O2S
Molecular Weight 410.572
Charge 0
Count
MOL RATIO 1 MOL RATIO (average)
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Description

Piperacetazine (Quide) is an antipsychotic prodrug, most notably used for schizophrenia. The study indicates that Quide is a useful addition to the armamentarium of the physician faced with the difficult problem of treating the chronic hospitalized patient with a schizophrenic illness. Side effects of the drug were generally mild, and there was no evidence that it would produce blood dyscrasias or liver impairment.

Originator

Approval Year

Conditions

ConditionModalityTargetsHighest PhaseProduct
Primary
QUIDE

PubMed

Sample Use Guides

In Vivo Use Guide
Unknown
Route of Administration: Oral
In Vitro Use Guide
Unknown
Substance Class Chemical
Record UNII
KL6248WNW4
Record Status Validated (UNII)
Record Version