U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
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Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:17:03 GMT 2025
Edited
by admin
on Tue Apr 01 17:17:03 GMT 2025
Protein Type ENZYME
Protein Sub Type SERINE/THREONINE-PROTEIN KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
J8URS97OQY
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 12
Common Name English
DLK
Preferred Name English
LEUCINE-ZIPPER PROTEIN KINASE
Common Name English
DUAL LEUCINE ZIPPER BEARING KINASE
Common Name English
ZPK
Common Name English
MAP3K12
Common Name English
MAPK-UPSTREAM KINASE
Common Name English
Code System Code Type Description
FDA UNII
J8URS97OQY
Created by admin on Tue Apr 01 17:17:03 GMT 2025 , Edited by admin on Tue Apr 01 17:17:03 GMT 2025
PRIMARY
UNIPROT
Q12852
Created by admin on Tue Apr 01 17:17:03 GMT 2025 , Edited by admin on Tue Apr 01 17:17:03 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_607] [1_695] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_37] [1_43] THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL